Compile Data Set for Download or QSAR
maximum 50k data
Found 17 of ki for monomerid = 50071754
TargetNeuromedin-B receptor(RAT)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi:  6.30nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi:  6.30nMAssay Description:Binding affinity against human NMB receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi:  6.30nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human NMB receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetBombesin(Frog)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin(Frog)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi:  127nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi:  134nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi:  174nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi:  180nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi:  248nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(RAT)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi:  340nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi:  4.80E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi:  7.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article