Affinity DataKi: 5.10nMAssay Description:Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Binding affinity to human cloned dopamine D4 receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Florida A&M University
Curated by ChEMBL
Florida A&M University
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Displacement [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 23.6nMAssay Description:Binding affinity to human cloned 5HT2A receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Florida A&M University
Curated by ChEMBL
Florida A&M University
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Displacement [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 43.3nMAssay Description:Binding affinity to human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Florida A&M University
Curated by ChEMBL
Florida A&M University
Curated by ChEMBL
Affinity DataKi: 56.6nMAssay Description:Binding affinity to human SERTMore data for this Ligand-Target Pair
Affinity DataKi: 117nMAssay Description:Binding affinity to human cloned 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 159nMAssay Description:Binding affinity to human cloned dopamine D3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 163nMAssay Description:Binding affinity to human cloned dopamine D1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 189nMAssay Description:Binding affinity to human cloned histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 296nMAssay Description:Binding affinity to human cloned 5HT6 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 495nMAssay Description:Binding affinity to human cloned 5HT2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 851nMAssay Description:Binding affinity to rat NETMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Florida A&M University
Curated by ChEMBL
Florida A&M University
Curated by ChEMBL
Affinity DataKi: 872nMAssay Description:Binding affinity to human cloned muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Florida A&M University
Curated by ChEMBL
Florida A&M University
Curated by ChEMBL
Affinity DataKi: 1.15E+3nMAssay Description:Binding affinity to human DATMore data for this Ligand-Target Pair
Affinity DataKi: 1.43E+3nMAssay Description:Binding affinity to human cloned 5HT2C receptorMore data for this Ligand-Target Pair