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TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM24566(JMC515449 Compound 1 | Wyeth 14,643 | 2-({4-chloro...)
Affinity DataKon:  2.30M-1s-1Assay Description:Binding affinity to PPARgamma (unknown origin) assessed as kinetic dissociation constant by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50235985(CHEMBL4092600)
Affinity DataKon:  0.0990M-1s-1Assay Description:Binding affinity to PPARgamma (unknown origin) assessed as kinetic dissociation constant by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50235986(CHEMBL4073499)
Affinity DataKon:  0.0950M-1s-1Assay Description:Binding affinity to PPARgamma (unknown origin) assessed as kinetic dissociation constant by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50030474(US9562012, rosiglitazone | CHEBI:50122 | Avandamet...)
Affinity DataKon:  0.145M-1s-1Assay Description:Binding affinity to PPARgamma (unknown origin) assessed as kinetic dissociation constant by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)