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Report error Found 135 of ki for UniProtKB: P13631
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataKi:  0.0400nMAssay Description:Agonistic activity towards retinoic acid receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of [3H]RA to binding Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In DepthDetails Article

TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity towards human Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article

TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataKi:  0.700nMAssay Description:Binding affinity against Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha [200-419]/gamma [183-417](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM36811(BMS614)
Affinity DataKi:  1nM ΔG°:  -11.4kcal/molepH: 8.0 T: 2°CAssay Description:Competitive assay were perform with 5nM tritiated all-trans retinoic acid (t-RA; 5nM) with or without 100-fold excess of non-radioactive t-RA (500nM)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRetinoic acid receptor alpha [200-419]/gamma [183-417](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM36810(BMS753 | US9963439, BMS753)
Affinity DataKi:  1nM ΔG°:  -11.4kcal/molepH: 8.0 T: 2°CAssay Description:Competitive assay were perform with 5nM tritiated all-trans retinoic acid (t-RA; 5nM) with or without 100-fold excess of non-radioactive t-RA (500nM)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM31892(CHEMBL705 | 9-cis retinoic acid | alitretinoin | P...)
Affinity DataKi:  1nMAssay Description:Agonistic activity towards retinoic acid receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma [183-417](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM31889(BMS 961 | BMS961 | BMS270394)
Affinity DataKi:  1.5nM ΔG°:  -11.2kcal/molepH: 8.0 T: 2°CAssay Description:Competitive assay were perform with 5nM tritiated all-trans retinoic acid (t-RA; 5nM) with or without 100-fold excess of non-radioactive t-RA (500nM)...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048296(4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-anthrace...)
Affinity DataKi:  2nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataKi:  3nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50032219(4-[(E)-2-(5,6,7,8-tetrahydro-5,5,8,8-tetramethyl-2...)
Affinity DataKi:  5nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048295(4-[(E)-2-(3-tert-Butyl-4-methoxy-phenyl)-propenyl]...)
Affinity DataKi:  13nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataKi:  19nMAssay Description:Inhibition of [3H]ATRA binding to Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50290081(3-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-naphthal...)
Affinity DataKi:  19nMAssay Description:Binding affinity towards Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article

TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048278(4-[(E)-2-(3-Adamantan-1-yl-4-hydroxy-phenyl)-vinyl...)
Affinity DataKi:  20nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM31892(CHEMBL705 | 9-cis retinoic acid | alitretinoin | P...)
Affinity DataKi:  20nMAssay Description:Inhibition of [3H]ATRA binding to Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048293(4-{(E)-2-[4-Hydroxy-3-(1-methyl-cyclohexyl)-phenyl...)
Affinity DataKi:  27nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048285(4-{(E)-2-[4-Methoxy-3-(1-methyl-cyclohexyl)-phenyl...)
Affinity DataKi:  29nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50290137((2E,4E)-3-Methyl-5-{2-[(E)-2-(3,3,6,6-tetramethyl-...)
Affinity DataKi:  32nMAssay Description:Binding affinity towards human Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article

TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048289(6-[3-Adamantan-1-yl-4-(2,3-dihydroxy-propyl)-pheny...)
Affinity DataKi:  34nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048281(6-(5',6',7',8'-tetrahydro-5',5',8',8'-tetramethyl-...)
Affinity DataKi:  40nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048281(6-(5',6',7',8'-tetrahydro-5',5',8',8'-tetramethyl-...)
Affinity DataKi:  40nMAssay Description:Binding affinity towards Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article

TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048276(4-[(E)-2-(3-Adamantan-1-yl-4-hydroxy-phenyl)-prope...)
Affinity DataKi:  53nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048284(6-[3-Adamantan-1-yl-4-(3-hydroxy-propyl)-phenyl]-n...)
Affinity DataKi:  72nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048291(6-[3'-(1-adamantyl)-4'-hydroxyphenyl]-2-naphthalen...)
Affinity DataKi:  77nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048290(4-[(E)-2-(3-tert-Butyl-4-hydroxy-phenyl)-propenyl]...)
Affinity DataKi:  85nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048277(4-[(E)-2-(3-Adamantan-1-yl-4-methoxy-phenyl)-prope...)
Affinity DataKi:  95nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048287(6-[4-Hydroxy-3-(1-methyl-cyclohexyl)-phenyl]-napht...)
Affinity DataKi:  121nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50052033((2E,4E,6E)-7-(3,5-Di-tert-butyl-phenyl)-3-methyl-o...)
Affinity DataKi:  124nMAssay Description:Inhibition of [3H]ATRA binding to Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50052033((2E,4E,6E)-7-(3,5-Di-tert-butyl-phenyl)-3-methyl-o...)
Affinity DataKi:  124nMAssay Description:Inhibition of [3H]ATRA binding to Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048280(6-(3-adamantan-1-yl-4-methoxyphenyl)naphthalene-2-...)
Affinity DataKi:  130nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi:  130nMAssay Description:Selective activity towards retinoic acid receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048280(6-(3-adamantan-1-yl-4-methoxyphenyl)naphthalene-2-...)
Affinity DataKi:  130nMAssay Description:Binding affinity towards Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article

TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50290078(3-(3-Adamantan-1-yl-4-hydroxy-phenyl)-2H-chromene-...)
Affinity DataKi:  148nMAssay Description:Binding affinity towards Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article

TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048297(6-[3-Adamantan-1-yl-4-(2,3-dihydroxy-propoxy)-phen...)
Affinity DataKi:  151nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048282(6-[3-Adamantan-1-yl-4-(1,2-dihydroxy-ethyl)-phenyl...)
Affinity DataKi:  153nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048292(6-[4-Methoxy-3-(1-methyl-cyclohexyl)-phenyl]-napht...)
Affinity DataKi:  160nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50290082(3-(3-Adamantan-1-yl-4-methoxy-phenyl)-2H-chromene-...)
Affinity DataKi:  174nMAssay Description:Binding affinity towards Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article

TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048294(6-(3-tert-Butyl-4-hydroxy-phenyl)-naphthalene-2-ca...)
Affinity DataKi:  200nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048294(6-(3-tert-Butyl-4-hydroxy-phenyl)-naphthalene-2-ca...)
Affinity DataKi:  200nMAssay Description:Binding affinity towards Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article

TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50283073(6-[(2E,4E,6E,8E)-3,7-Dimethyl-9-(2,6,6-trimethyl-c...)
Affinity DataKi:  280nMAssay Description:Inhibition of [3H]RA binding to Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In DepthDetails Article

TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048283(6-(3-Adamantan-1-yl-4-hydroxymethyl-phenyl)-naphth...)
Affinity DataKi:  386nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50092055(CHEMBL7301 | N-(4-hydroxyphenyl)-retinamide | 4-hy...)
Affinity DataKi: >400nMAssay Description:Binding affinity against Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048279(6-(3-tert-Butyl-4-methoxy-phenyl)-naphthalene-2-ca...)
Affinity DataKi:  426nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50052588((2E,4E,6Z)-7-(3-Methoxy-5,5,8,8-tetramethyl-5,6,7,...)
Affinity DataKi:  437nMAssay Description:Inhibition of [3H]ATRA binding to Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061615(4-(10,10,13,13,15-Pentamethyl-11,12,13,15-tetrahyd...)
Affinity DataKi:  490nMAssay Description:Antagonistic activity towards retinoic acid receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50290083(3-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-2H-chromene...)
Affinity DataKi:  531nMAssay Description:Binding affinity towards Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article

TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50283072((2E,4E,6E,8E)-3,7-Dimethyl-9-(2,6,6-trimethyl-cycl...)
Affinity DataKi:  710nMAssay Description:Inhibition of [3H]RA to binding Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
In DepthDetails Article

TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50048298(6-(4,4-Dimethyl-chroman-6-yl)-naphthalene-2-carbox...)
Affinity DataKi:  860nMAssay Description:Binding affinity to retinoic acid receptor (RAR) gamma using [3H]CD 367 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50033079(4-[1-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-napht...)
Affinity DataKi:  887nMAssay Description:Inhibition of [3H]ATRA binding to RAR gamma receptorMore data for this Ligand-Target Pair
In DepthDetails Article

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