Compile Data Set for Download or QSAR
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Found 10 of ki for UniProtKB: P68403
TargetProtein kinase C beta type(Rattus norvegicus (rat))
University of California San Diego

LigandPNGBDBM3149(2-{[2,6-dihydroxy-4-({[(3R,4R)-3-[(4-hydroxybenzen...)
Affinity DataKi:  5.30nM ΔG°:  -11.5kcal/moleT: 2°CAssay Description:Protein kinase C (PKC) enzyme inhibition assay using purified rat brain protein kinase C from Calbiochem #539494.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Rattus norvegicus (rat))
University of California San Diego

LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataKi:  19nM ΔG°:  -10.7kcal/moleT: 2°CAssay Description:Protein kinase C (PKC) enzyme inhibition assay using purified rat brain protein kinase C from Calbiochem #539494.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Rattus norvegicus (rat))
University of California San Diego

LigandPNGBDBM36604(5'-Deoxybalanol, 7)
Affinity DataKi:  69nM ΔG°:  -9.93kcal/mole IC50:  95nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC) enzyme inhibition assay using purified rat brain protein kinase C from Calbiochem #539494.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Rattus norvegicus (rat))
University of California San Diego

LigandPNGBDBM36603(4'',6''-Dideoxybalanol, 6)
Affinity DataKi:  80nM ΔG°:  -9.84kcal/mole IC50:  111nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC) enzyme inhibition assay using purified rat brain protein kinase C from Calbiochem #539494.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Rattus norvegicus (rat))
University of California San Diego

LigandPNGBDBM3207(10''-Deoxybalanol, 4 | 2-{[2,6-dihydroxy-4-({[(3R,...)
Affinity DataKi:  640nM ΔG°:  -8.59kcal/mole IC50:  834nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC) enzyme inhibition assay using purified rat brain protein kinase C from Calbiochem #539494.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Rattus norvegicus (rat))
University of California San Diego

LigandPNGBDBM36605(KT5720, 9)
Affinity DataKi: >2.00E+3nM ΔG°: >-7.90kcal/moleT: 2°CAssay Description:Protein kinase C (PKC) enzyme inhibition assay using purified rat brain protein kinase C from Calbiochem #539494.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Rattus norvegicus (rat))
University of California San Diego

LigandPNGBDBM36602(14''-Decarboxybalanol hydrochloride, 5)
Affinity DataKi:  5.00E+3nM ΔG°:  -7.35kcal/mole IC50:  6.90E+3nMT: 2°CAssay Description:Protein kinase C (PKC) enzyme inhibition assay using purified rat brain protein kinase C from Calbiochem #539494.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Rattus norvegicus (rat))
University of California San Diego

LigandPNGBDBM36606(H-89, 10)
Affinity DataKi:  3.17E+4nM ΔG°:  -6.24kcal/moleT: 2°CAssay Description:Protein kinase C (PKC) enzyme inhibition assay using purified rat brain protein kinase C from Calbiochem #539494.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Rattus norvegicus (rat))
University of California San Diego

LigandPNGBDBM36601(Hexahydroazepine, 3)
Affinity DataKi: >1.00E+6nM ΔG°: >-4.16kcal/moleT: 2°CAssay Description:Protein kinase C (PKC) enzyme inhibition assay using purified rat brain protein kinase C from Calbiochem #539494.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Rattus norvegicus (rat))
University of California San Diego

LigandPNGBDBM36600(Benzophenone fragment, 2)
Affinity DataKi: >1.00E+6nM ΔG°: >-4.16kcal/molepH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC) enzyme inhibition assay using purified rat brain protein kinase C from Calbiochem #539494.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed