TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Affinity towards Alpha-1A adrenergic receptor in membranes from bovine frontal cortex using [3H]-prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Affinity towards Alpha-1A adrenergic receptor in membranes from bovine frontal cortex using [3H]-prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 0.820nMAssay Description:Affinity towards Alpha-1A adrenergic receptor in membranes from bovine frontal cortex using [3H]-prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Affinity towards Alpha-1A adrenergic receptor in membranes from bovine frontal cortex using [3H]-prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Affinity towards Alpha-1A adrenergic receptor in membranes from bovine frontal cortex using [3H]-prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Affinity towards Alpha-1A adrenergic receptor in membranes from bovine frontal cortex using [3H]-prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Binding affinity was tested on cloned bovine Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Affinity towards Alpha-1A adrenergic receptor in membranes from bovine frontal cortex using [3H]-prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Affinity towards Alpha-1A adrenergic receptor in membranes from bovine frontal cortex using [3H]-prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Affinity towards Alpha-1A adrenergic receptor in membranes from bovine frontal cortex using [3H]-prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Affinity towards Alpha-1A adrenergic receptor in membranes from bovine frontal cortex using [3H]-prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Affinity towards Alpha-1A adrenergic receptor in membranes from bovine frontal cortex using [3H]-prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Affinity towards Alpha-1A adrenergic receptor in membranes from bovine frontal cortex using [3H]-prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 85nMAssay Description:Affinity towards Alpha-1A adrenergic receptor in membranes from bovine frontal cortex using [3H]-prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Affinity towards Alpha-1A adrenergic receptor in membranes from bovine frontal cortex using [3H]-prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Compound was evaluated for binding affinity at bovine brain Alpha-1 adrenergic receptor in a filtration-based assay using [3H]prazosin as the radioli...More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Affinity towards Alpha-1A adrenergic receptor in membranes from bovine frontal cortex using [3H]-prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Affinity towards Alpha-1A adrenergic receptor in membranes from bovine frontal cortex using [3H]-prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Affinity towards Alpha-1A adrenergic receptor in membranes from bovine frontal cortex using [3H]-prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Affinity towards Alpha-1A adrenergic receptor in membranes from bovine frontal cortex using [3H]-prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Compound was evaluated for binding affinity at bovine brain Alpha-1 adrenergic receptor in a filtration-based assay using [3H]prazosin as the radioli...More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Compound was evaluated for binding affinity at bovine brain Alpha-1 adrenergic receptor determined in a filtration-based assay using [3H]prazosin as ...More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 950nMAssay Description:Binding affinity was tested on cloned bovine Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was evaluated for binding affinity at bovine brain Alpha-1 adrenergic receptor in a filtration-based assay using [3H]prazosin as the radioli...More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Compound was evaluated for binding affinity at bovine brain Alpha-1 adrenergic receptor in a filtration-based assay using [3H]prazosin as the radioli...More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Compound was evaluated for binding affinity at bovine brain Alpha-1 adrenergic receptor in a filtration-based assay using [3H]prazosin as the radioli...More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Compound was evaluated for binding affinity at bovine brain Alpha-1 adrenergic receptor in a filtration-based assay using [3H]prazosin as the radioli...More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair