Compile Data Set for Download or QSAR
maximum 50k data
Found 23 of ic50 for UniProtKB: P52500
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112639(CHEMBL402688 | pQ-Q-R-Y-G-N-Q-W-A-V-G-H-L-M-NH2)
Affinity DataIC50:  1.10nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112626(CHEMBL442514 | Carbocyanine derivative)
Affinity DataIC50:  1.80nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112623((FITC-Q-W-A-V-G-H-L-M-NH2) | CHEMBL274327)
Affinity DataIC50:  3.20nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112643((DTPA-P-Q-R-Y-G-N-Q-W-A-V-G-H-L-M-NH2) | CHEMBL442...)
Affinity DataIC50:  4.70nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112611((K-G-S-G-Q-W-A-V-G-H-L-M-NH2) | CHEMBL405669)
Affinity DataIC50:  4.80nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112640((epsilon-DTPA-K-Q-W-A-V-G-H-L-M-NH2) | CHEMBL21696...)
Affinity DataIC50:  4.80nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112629((epsilon-FITC-K-Q-W-A-V-G-H-L-M-NH2) | CHEMBL38528...)
Affinity DataIC50:  5.70nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112632((alpha-FITC-K-Q-W-A-V-G-H-L-M-NH2) | CHEMBL428280)
Affinity DataIC50:  5.80nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112619((G-S-G-Q-W-A-V-G-H-L-M-NH2) | CHEMBL408739)
Affinity DataIC50:  7.60nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112633((FITC-G-S-G-Q-W-A-V-G-H-L-M-NH2) | CHEMBL385928)
Affinity DataIC50:  9.20nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112635((alpha,epsilon-(-FITC)2-K-Q-W-A-V-G-H-L-M-NH2) | C...)
Affinity DataIC50:  9.5nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112620((epsilon-FITC-K-G-S-G-Q-W-A-V-G-H-L-M-NH2) | CHEMB...)
Affinity DataIC50:  9.60nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112625((K-Q-W-A-V-G-H-L-M-NH2) | CHEMBL269310)
Affinity DataIC50:  10.5nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112627((alpha-FITC-epsilon-DOTA-K-Q-W-A-V-G-H-L-M-NH2) | ...)
Affinity DataIC50:  15nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112646((alpha-FITC-K-G-S-G-Q-W-A-V-G-H-L-M-NH2) | CHEMBL4...)
Affinity DataIC50:  15.6nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112614((alpha-FITC-epsilon-DTPA-K-Q-W-A-V-G-H-L-M-NH2) | ...)
Affinity DataIC50:  20nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112616((alpha,epsilon-(FITC)2-K-G-S-G-Q-W-A-V-G-H-L-M-NH2...)
Affinity DataIC50:  20.5nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112642((Q-W-A-V-G-H-L-M-NH2) | CHEMBL300318)
Affinity DataIC50:  28.3nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112630((alpha,epsilon-(DTPA)2-K-Q-W-A-V-G-H-L-M-NH2) | CH...)
Affinity DataIC50:  240nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112621((alpha-DTPA-epsilon-FITC-K-Q-W-A-V-G-H-L-M-NH2) | ...)
Affinity DataIC50:  276nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112622((alpha-DTPA-K-Q-W-A-V-G-H-L-M-NH2) | CHEMBL440609)
Affinity DataIC50:  410nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50280413(5'-bromo-1'-(3,4-dichlorobenzyl)spiro[tetrahydro-1...)
Affinity DataIC50:  1.50E+3nMAssay Description:Compound was evaluated for displacement of radiolabelled [I-125]GRP from rat brain receptor; 1.5-3 microMMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50280412(2-{3-[1-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-meth-...)
Affinity DataIC50:  1.50E+3nMAssay Description:Compound was evaluated for displacement of radiolabelled [I-125]GRP from rat brain receptor; 1.5-3 microMMore data for this Ligand-Target Pair
In DepthDetails Article