TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.00500nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma 1 receptor in guinea pig brain microsomesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.00500nMAssay Description:Displacement of (+)-[3H]-pentazocine from sigma 1 receptor in guinea pig whole brain microsomesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.00500nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pigMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.0110nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma 1 receptor in guinea pig liver microsomesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.0110nMAssay Description:Displacement of (+)-[3H]-pentazocine from sigma 1 receptor in guinea pig liver microsomesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.0300nMAssay Description:Displacement of [3H]-pentazocine from sigma 1 receptor in guinea pig brain membrane after 120 minsMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.0300nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.0360nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.0500nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.0700nMAssay Description:Displacement of (+)-[3H]pentazocine from guinea pig brain membrane sigma1 receptor by scintillation spectrometric methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.0800nMAssay Description:Displacement of (+)-[3H]-pentazocine from recombinant guinea pig His6-tagged sigma 1 receptor expressed in Saccharomyces cerevisiae WAO microsomesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.0800nMAssay Description:The compound was tested for inhibition of [3H]-5-hydroxy tryptamine uptake in HEK cells by expressing cDNA for human tryptamine transporterMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.110nMAssay Description:Displacement of [3H]-pentazocine from sigma 1 receptor in guinea pig brain membrane after 120 minsMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.110nMAssay Description:Displacement of [3H](+)-pentazocine ((+)-[2S-(2R,6R,11R)]-1,2,3,4,5,6-hexahydro-6,11-dimethyl- 3-(3-methyl-2-butenyl)-2,6-methano-3-benzazocine- 8-ol...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.120nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in Dunkin guinea pig brain membrane without cerebellumMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.140nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membranes without cerebellumMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.140nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.140nMAssay Description:Binding affinity against human progesterone receptor (hPR) in a competitive binding assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.152nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane by solid scintillation analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.194nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain homogenate incubated for 150 mins by liquid scintillation counting meth...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]-(+)-pentazocin from sigma1 receptor in guinea pig brain P2 membranes after 120 minsMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes by microbeta scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.210nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membranes without cerebellumMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.220nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.220nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.240nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H](+)-pentazocine ((+)-[2S-(2R,6R,11R)]-1,2,3,4,5,6-hexahydro-6,11-dimethyl- 3-(3-methyl-2-butenyl)-2,6-methano-3-benzazocine- 8-ol...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of (+)-[3H]pentazocine from guinea pig brain membrane sigma1 receptor by scintillation spectrometric methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.260nMAssay Description:Inhibition of purified human kidney thiopurine methyltransferase (TPMT)More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in Dunkin-Hartley guinea pig brain membranes incubated for 180 mins by liquid scintillatio...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.290nMAssay Description:Displacement of [3H]-(+)pentazocine from guinea pig brain sigma 1-type opioid receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.290nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.290nMAssay Description:Displacement of (+)-[3H]pentazocine from guinea pig brain membrane sigma1 receptor by scintillation spectrometric methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]-(+)pentazocine from sigma-1 receptor in guinea pig brain membranes after 180 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:The affinity of test compounds at sigma-1 and sigma-2 receptors was also determined by displacement of different known labeled sigma-2 or sigma-1 lig...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma 1 receptor in guinea pig liver homogenates after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain cortex membranes measured after 120 mins by scintillation counting meth...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.310nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain cortex membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.310nMAssay Description:Displacement of [3H]-(+)pentazocine from guinea pig brain sigma 1-type opioid receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.320nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain cortex membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.320nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair