TargetGhrelin O-acyltransferase(Mus musculus)
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataIC50: 3.10nMAssay Description:Inhibition of mouse GOAT expressed in baculovirus infected sf9 insect cell microsomes using biotinylated des-acyl ghrelin and octanoyl-CoA -CoA as su...More data for this Ligand-Target Pair
TargetGhrelin O-acyltransferase(Mus musculus)
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataIC50: 3.30nMAssay Description:Inhibition of mouse GOAT expressed in baculovirus infected sf9 insect cell microsomes using biotinylated des-acyl ghrelin and octanoyl-CoA -CoA as su...More data for this Ligand-Target Pair
TargetGhrelin O-acyltransferase(Mus musculus)
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co...More data for this Ligand-Target Pair
TargetGhrelin O-acyltransferase(Mus musculus)
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co...More data for this Ligand-Target Pair
TargetGhrelin O-acyltransferase(Mus musculus)
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co...More data for this Ligand-Target Pair
TargetGhrelin O-acyltransferase(Mus musculus)
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataIC50: 7.50E+3nMAssay Description:Antagonist activity at mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using ghrelin(1 to 5) pentapeptide as substrate preincub...More data for this Ligand-Target Pair
TargetGhrelin O-acyltransferase(Mus musculus)
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Antagonist activity at mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using ghrelin(1 to 5) pentapeptide as substrate preincub...More data for this Ligand-Target Pair
TargetGhrelin O-acyltransferase(Mus musculus)
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co...More data for this Ligand-Target Pair
TargetGhrelin O-acyltransferase(Mus musculus)
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co...More data for this Ligand-Target Pair
TargetGhrelin O-acyltransferase(Mus musculus)
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co...More data for this Ligand-Target Pair