Compile Data Set for Download or QSAR
maximum 50k data
Found 106 of ec50 for UniProtKB: Q5NUL3
TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50408138(CHEMBL5286838)
Affinity DataEC50:  5.30nMAssay Description:Antagonist effect against 2-methyl-5-HT activity at 5-HT3 receptor in longitudinal muscle myenteric plexus from guinea pig ileumMore data for this Ligand-Target Pair
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50543524(CHEMBL4637969)
Affinity DataEC50:  6nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50543530(CHEMBL4646784)
Affinity DataEC50:  6nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50543525(CHEMBL4639009)
Affinity DataEC50:  45nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM382131(4-(4-((2-(5,6,7,8-tetrahydronaphthalen-2-yl)cycloh...)
Affinity DataEC50:  50nMAssay Description:Antagonist effect against 2-methyl-5-HT activity at 5-HT3 receptor in longitudinal muscle myenteric plexus from guinea pig ileumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50408139(CHEMBL5272316)
Affinity DataEC50:  50nMAssay Description:Antagonist effect against 2-methyl-5-HT activity at 5-HT3 receptor in longitudinal muscle myenteric plexus from guinea pig ileumMore data for this Ligand-Target Pair
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM382129(4-(4-((4'-cyclopropyl-3,4,5,6-tetrahydro-[1,1'-bip...)
Affinity DataEC50:  50nMAssay Description:Antagonist effect against 2-methyl-5-HT activity at 5-HT3 receptor in longitudinal muscle myenteric plexus from guinea pig ileumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM382129(4-(4-((4'-cyclopropyl-3,4,5,6-tetrahydro-[1,1'-bip...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at FFA4 (unknown origin) expressed in CHO-K1 cells by BRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM382129(4-(4-((4'-cyclopropyl-3,4,5,6-tetrahydro-[1,1'-bip...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50408138(CHEMBL5286838)
Affinity DataEC50:  60nMAssay Description:Antagonist effect against 2-methyl-5-HT activity at 5-HT3 receptor in longitudinal muscle myenteric plexus from guinea pig ileumMore data for this Ligand-Target Pair
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50543526(CHEMBL4646553)
Affinity DataEC50:  61nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50543519(CHEMBL4642324)
Affinity DataEC50:  71nMAssay Description:Modulation of GPR120 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50543528(CHEMBL4638249)
Affinity DataEC50:  110nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50408138(CHEMBL5286838)
Affinity DataEC50:  120nMAssay Description:Antagonist effect against 2-methyl-5-HT activity at 5-HT3 receptor in longitudinal muscle myenteric plexus from guinea pig ileumMore data for this Ligand-Target Pair
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50408137(CHEMBL5275980)
Affinity DataEC50:  125nMAssay Description:Antagonist effect against 2-methyl-5-HT activity at 5-HT3 receptor in longitudinal muscle myenteric plexus from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50610009(CHEMBL5266881)
Affinity DataEC50:  150nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50609986(CHEMBL5290885)
Affinity DataEC50:  150nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50420167(CHEMBL2058533)
Affinity DataEC50:  158nMAssay Description:Agonist activity at human FFA4 receptor expressed in CHO-K1 cells assessed as increase in amplitude of dynamic mass redistribution response by DMR as...More data for this Ligand-Target Pair
TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50408137(CHEMBL5275980)
Affinity DataEC50:  165nMAssay Description:Antagonist effect against 2-methyl-5-HT activity at 5-HT3 receptor in longitudinal muscle myenteric plexus from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50543527(CHEMBL4647832)
Affinity DataEC50:  179nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50543523(CHEMBL4642294)
Affinity DataEC50:  220nMAssay Description:Modulation of GPR120 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50543523(CHEMBL4642294)
Affinity DataEC50:  220nMAssay Description:Agonist activity at human GPR120 expressed in CHO cells assessed as intracellular phosphorylated ERK incubated for 16 to 18 hrs by AlphaScreen SureFi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50543529(CHEMBL4641735)
Affinity DataEC50:  270nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50609987(CHEMBL5278642)
Affinity DataEC50:  360nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50609991(CHEMBL5273250)
Affinity DataEC50:  560nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50609998(CHEMBL5278718)
Affinity DataEC50:  590nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50610010(CHEMBL5268316)
Affinity DataEC50:  600nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50610007(CHEMBL5287642)
Affinity DataEC50:  600nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50609989(CHEMBL5268389)
Affinity DataEC50:  600nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50610054(CHEMBL5266170)
Affinity DataEC50:  640nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50610006(CHEMBL5281423)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50609983(CHEMBL5276740)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50609980(CHEMBL5284985)
Affinity DataEC50:  1.21E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50609990(CHEMBL5286544)
Affinity DataEC50:  1.27E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50609994(CHEMBL5272492)
Affinity DataEC50:  1.32E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50554587(CHEMBL4794951)
Affinity DataEC50:  1.55E+3nMAssay Description:Agonist activity at human FFA4 receptor expressed in CHO-K1 cells assessed as increase in amplitude of dynamic mass redistribution response by DMR as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50609996(CHEMBL5289099)
Affinity DataEC50:  1.57E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50610042(CHEMBL5285139)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50554598(CHEMBL4744629)
Affinity DataEC50:  2.19E+3nMAssay Description:Agonist activity at human FFA4 receptor expressed in CHO-K1 cells assessed as increase in amplitude of dynamic mass redistribution response by DMR as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50610055(CHEMBL5278789)
Affinity DataEC50:  2.19E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50610027(CHEMBL5268800)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50610003(CHEMBL5289929)
Affinity DataEC50:  3.03E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM22496(3-(4-{[(3-phenoxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50:  3.16E+3nMAssay Description:Agonist activity at human FFA4 expressed in HEK293 cells assessed as stimulation of intracellular calcium mobilization measured at every 1 secs for 6...More data for this Ligand-Target Pair
TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM22496(3-(4-{[(3-phenoxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50:  3.50E+3nMAssay Description:Antagonist effect against 2-methyl-5-HT activity at 5-HT3 receptor in longitudinal muscle myenteric plexus from guinea pig ileumMore data for this Ligand-Target Pair
TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50554596(CHEMBL4791789)
Affinity DataEC50:  3.55E+3nMAssay Description:Agonist activity at human FFA4 receptor expressed in CHO-K1 cells assessed as increase in amplitude of dynamic mass redistribution response by DMR as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50554597(CHEMBL4743951)
Affinity DataEC50:  3.98E+3nMAssay Description:Agonist activity at human FFA4 receptor expressed in CHO-K1 cells assessed as increase in amplitude of dynamic mass redistribution response by DMR as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50610038(CHEMBL5273939)
Affinity DataEC50:  4.00E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50609993(CHEMBL5289774)
Affinity DataEC50:  4.39E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50554588(CHEMBL4795755)
Affinity DataEC50:  4.90E+3nMAssay Description:Agonist activity at human FFA4 receptor expressed in CHO-K1 cells assessed as increase in amplitude of dynamic mass redistribution response by DMR as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)TBA
LigandPNGBDBM50610034(CHEMBL5268182)
Affinity DataEC50:  5.00E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
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