Affinity DataEC50: 5.30nMAssay Description:Antagonist effect against 2-methyl-5-HT activity at 5-HT3 receptor in longitudinal muscle myenteric plexus from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 45nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Antagonist effect against 2-methyl-5-HT activity at 5-HT3 receptor in longitudinal muscle myenteric plexus from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Antagonist effect against 2-methyl-5-HT activity at 5-HT3 receptor in longitudinal muscle myenteric plexus from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Antagonist effect against 2-methyl-5-HT activity at 5-HT3 receptor in longitudinal muscle myenteric plexus from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist activity at FFA4 (unknown origin) expressed in CHO-K1 cells by BRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 60nMAssay Description:Antagonist effect against 2-methyl-5-HT activity at 5-HT3 receptor in longitudinal muscle myenteric plexus from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 61nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 71nMAssay Description:Modulation of GPR120 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 110nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:Antagonist effect against 2-methyl-5-HT activity at 5-HT3 receptor in longitudinal muscle myenteric plexus from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 125nMAssay Description:Antagonist effect against 2-methyl-5-HT activity at 5-HT3 receptor in longitudinal muscle myenteric plexus from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 150nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 150nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 158nMAssay Description:Agonist activity at human FFA4 receptor expressed in CHO-K1 cells assessed as increase in amplitude of dynamic mass redistribution response by DMR as...More data for this Ligand-Target Pair
Affinity DataEC50: 165nMAssay Description:Antagonist effect against 2-methyl-5-HT activity at 5-HT3 receptor in longitudinal muscle myenteric plexus from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 179nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 220nMAssay Description:Modulation of GPR120 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 220nMAssay Description:Agonist activity at human GPR120 expressed in CHO cells assessed as intracellular phosphorylated ERK incubated for 16 to 18 hrs by AlphaScreen SureFi...More data for this Ligand-Target Pair
Affinity DataEC50: 270nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 360nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 560nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 590nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 600nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 600nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 600nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 640nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 1.20E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 1.20E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 1.21E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 1.27E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 1.32E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 1.55E+3nMAssay Description:Agonist activity at human FFA4 receptor expressed in CHO-K1 cells assessed as increase in amplitude of dynamic mass redistribution response by DMR as...More data for this Ligand-Target Pair
Affinity DataEC50: 1.57E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 2.00E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 2.19E+3nMAssay Description:Agonist activity at human FFA4 receptor expressed in CHO-K1 cells assessed as increase in amplitude of dynamic mass redistribution response by DMR as...More data for this Ligand-Target Pair
Affinity DataEC50: 2.19E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 3.00E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 3.03E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 3.16E+3nMAssay Description:Agonist activity at human FFA4 expressed in HEK293 cells assessed as stimulation of intracellular calcium mobilization measured at every 1 secs for 6...More data for this Ligand-Target Pair
Affinity DataEC50: 3.50E+3nMAssay Description:Antagonist effect against 2-methyl-5-HT activity at 5-HT3 receptor in longitudinal muscle myenteric plexus from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 3.55E+3nMAssay Description:Agonist activity at human FFA4 receptor expressed in CHO-K1 cells assessed as increase in amplitude of dynamic mass redistribution response by DMR as...More data for this Ligand-Target Pair
Affinity DataEC50: 3.98E+3nMAssay Description:Agonist activity at human FFA4 receptor expressed in CHO-K1 cells assessed as increase in amplitude of dynamic mass redistribution response by DMR as...More data for this Ligand-Target Pair
Affinity DataEC50: 4.00E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 4.39E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 4.90E+3nMAssay Description:Agonist activity at human FFA4 receptor expressed in CHO-K1 cells assessed as increase in amplitude of dynamic mass redistribution response by DMR as...More data for this Ligand-Target Pair
Affinity DataEC50: 5.00E+3nMAssay Description:Agonist activity at N-terminal FLAG tagged human FFAR4 transfected in African green monkey COS-7 cells assessed as accumulation of inositol phosphate...More data for this Ligand-Target Pair
Ligand Info