Compile Data Set for Download or QSAR
maximum 50k data
Found 31 of ec50 data for polymerid = 50001025,50007714
TargetMajor prion protein(Homo sapiens (Human))
Institut F£R Molekularbiologie Und Biophysik

Curated by ChEMBL
LigandPNGBDBM50015214(6-chloro-2-methoxy-9-acridinyl(4-diethylamino-1-me...)
Affinity DataEC50:  300nMAssay Description:Half maximal inhibition of Prion protein PrPsc formation was assayed in ScN2a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Homo sapiens (Human))
Institut F£R Molekularbiologie Und Biophysik

Curated by ChEMBL
LigandPNGBDBM50001888((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...)
Affinity DataEC50:  2.00E+3nMAssay Description:Half maximal inhibition of Prion protein PrPsc formation was assayed in ScN2a cellsMore data for this Ligand-Target Pair
TargetMajor prion protein(Homo sapiens (Human))
Institut F£R Molekularbiologie Und Biophysik

Curated by ChEMBL
LigandPNGBDBM22985(Aralen | CHEMBL76 | CHLOROQUINE PHOSPHATE | Chloro...)
Affinity DataEC50:  4.00E+3nMAssay Description:Half maximal inhibition of Prion protein PrPsc formation was assayed in ScN2a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Homo sapiens (Human))
Institut F£R Molekularbiologie Und Biophysik

Curated by ChEMBL
LigandPNGBDBM67545(N,N-dimethyl-3-(10-phenothiazinyl)-1-propanamine;h...)
Affinity DataEC50:  5.00E+3nMAssay Description:Half maximal inhibition of Prion protein PrPsc formation was assayed in ScN2a cellsMore data for this Ligand-Target Pair
TargetMajor prion protein(Homo sapiens (Human))
Institut F£R Molekularbiologie Und Biophysik

Curated by ChEMBL
LigandPNGBDBM50131719(CHEMBL39560 | acepromazine)
Affinity DataEC50:  5.00E+3nMAssay Description:Half maximal inhibition of Prion protein PrPsc formation was assayed in ScN2a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Mesocricetus auratus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50451083(CHEMBL1429474)
Affinity DataEC50:  7.02E+3nMAssay Description:Binding affinity to Syrian hamster PrPC assessed as inhibition of PrPC protein conversion to PrPSc by Western blotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Mesocricetus auratus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50451084(CHEMBL1631214)
Affinity DataEC50:  7.16E+3nMAssay Description:Binding affinity to Syrian hamster PrPC assessed as inhibition of PrPC protein conversion to PrPSc by Western blotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Mesocricetus auratus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50451087(CHEMBL1631213)
Affinity DataEC50:  7.17E+3nMAssay Description:Binding affinity to Syrian hamster PrPC assessed as inhibition of PrPC protein conversion to PrPSc by Western blotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Mesocricetus auratus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50451088(CHEMBL4215683)
Affinity DataEC50:  7.17E+3nMAssay Description:Binding affinity to Syrian hamster PrPC assessed as inhibition of PrPC protein conversion to PrPSc by Western blotMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMajor prion protein(Mesocricetus auratus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50451085(CHEMBL1631211)
Affinity DataEC50:  7.17E+3nMAssay Description:Binding affinity to Syrian hamster PrPC assessed as inhibition of PrPC protein conversion to PrPSc by Western blotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Mesocricetus auratus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50451086(CHEMBL4218996)
Affinity DataEC50:  7.17E+3nMAssay Description:Binding affinity to Syrian hamster PrPC assessed as inhibition of PrPC protein conversion to PrPSc by Western blotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Mesocricetus auratus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50451089(CHEMBL4206759)
Affinity DataEC50:  7.18E+3nMAssay Description:Binding affinity to Syrian hamster PrPC assessed as inhibition of PrPC protein conversion to PrPSc by Western blotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Mesocricetus auratus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50451090(CHEMBL1631209)
Affinity DataEC50:  7.18E+3nMAssay Description:Binding affinity to Syrian hamster PrPC assessed as inhibition of PrPC protein conversion to PrPSc by Western blotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Mesocricetus auratus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50451075(CHEMBL1311517)
Affinity DataEC50:  7.19E+3nMAssay Description:Binding affinity to Syrian hamster PrPC assessed as inhibition of PrPC protein conversion to PrPSc by Western blotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Mesocricetus auratus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50451091(CHEMBL1631206)
Affinity DataEC50:  7.20E+3nMAssay Description:Binding affinity to Syrian hamster PrPC assessed as inhibition of PrPC protein conversion to PrPSc by Western blotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Mesocricetus auratus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50451092(CHEMBL4215372)
Affinity DataEC50:  7.23E+3nMAssay Description:Binding affinity to Syrian hamster PrPC assessed as inhibition of PrPC protein conversion to PrPSc by Western blotMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMajor prion protein(Mesocricetus auratus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50451076(CHEMBL1418383)
Affinity DataEC50:  7.24E+3nMAssay Description:Binding affinity to Syrian hamster PrPC assessed as inhibition of PrPC protein conversion to PrPSc by Western blotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Mesocricetus auratus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50451093(CHEMBL4210951)
Affinity DataEC50:  7.24E+3nMAssay Description:Binding affinity to Syrian hamster PrPC assessed as inhibition of PrPC protein conversion to PrPSc by Western blotMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMajor prion protein(Mesocricetus auratus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50451095(CHEMBL1631123)
Affinity DataEC50:  7.24E+3nMAssay Description:Binding affinity to Syrian hamster PrPC assessed as inhibition of PrPC protein conversion to PrPSc by Western blotMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMajor prion protein(Mesocricetus auratus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50451079(CHEMBL4205700)
Affinity DataEC50:  7.25E+3nMAssay Description:Binding affinity to Syrian hamster PrPC assessed as inhibition of PrPC protein conversion to PrPSc by Western blotMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMajor prion protein(Mesocricetus auratus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50451077(CHEMBL4202679)
Affinity DataEC50:  7.27E+3nMAssay Description:Binding affinity to Syrian hamster PrPC assessed as inhibition of PrPC protein conversion to PrPSc by Western blotMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMajor prion protein(Mesocricetus auratus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50451078(CHEMBL1631117)
Affinity DataEC50:  7.29E+3nMAssay Description:Binding affinity to Syrian hamster PrPC assessed as inhibition of PrPC protein conversion to PrPSc by Western blotMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMajor prion protein(Mesocricetus auratus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50333113(8-methyl-7-(2-(piperidin-1-yl)ethylthio)-2,3-dihyd...)
Affinity DataEC50:  7.32E+3nMAssay Description:Binding affinity to Syrian hamster PrPC assessed as inhibition of PrPC protein conversion to PrPSc by Western blotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Mesocricetus auratus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50333112(3-amino-N-cyclopentyl-8-methylthieno[2,3-b]quinoli...)
Affinity DataEC50:  7.37E+3nMAssay Description:Binding affinity to Syrian hamster PrPC assessed as inhibition of PrPC protein conversion to PrPSc by Western blotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Mesocricetus auratus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50333111(2-(2-(butylamino)-1H-benzo[d]imidazol-1-yl)-1-(ind...)
Affinity DataEC50:  7.42E+3nMAssay Description:Binding affinity to Syrian hamster PrPC assessed as inhibition of PrPC protein conversion to PrPSc by Western blotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Mesocricetus auratus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50333110(CHEMBL1631113 | N-(1-(indolin-1-yl)-3-methyl-1-oxo...)
Affinity DataEC50:  7.43E+3nMAssay Description:Binding affinity to Syrian hamster PrPC assessed as inhibition of PrPC protein conversion to PrPSc by Western blotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Homo sapiens (Human))
Institut F£R Molekularbiologie Und Biophysik

Curated by ChEMBL
LigandPNGBDBM50017696((2-dimethylamino-2-methyl)ethyl-N-dibenzoparathiaz...)
Affinity DataEC50:  8.00E+3nMAssay Description:Half maximal inhibition of Prion protein PrPsc formation was assayed in ScN2a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Homo sapiens (Human))
Institut F£R Molekularbiologie Und Biophysik

Curated by ChEMBL
LigandPNGBDBM50131720(9,10-diazaanthracene | CHEMBL119870 | acridizine |...)
Affinity DataEC50: >1.00E+4nMAssay Description:Half maximal inhibition of Prion protein PrPsc formation was assayed in ScN2a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Homo sapiens (Human))
Institut F£R Molekularbiologie Und Biophysik

Curated by ChEMBL
LigandPNGBDBM50003659(5H-dibenzo[b,f]azepine-5-carboxamide | CARBAMAZEPI...)
Affinity DataEC50: >1.00E+4nMAssay Description:Half maximal inhibition of Prion protein PrPsc formation was assayed in ScN2a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Homo sapiens (Human))
Institut F£R Molekularbiologie Und Biophysik

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataEC50: >1.00E+4nMAssay Description:Half maximal inhibition of Prion protein PrPsc formation was assayed in ScN2a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Homo sapiens (Human))
Institut F£R Molekularbiologie Und Biophysik

Curated by ChEMBL
LigandPNGBDBM50010859(CHEMBL11 | IMIPRAMINE HYDROCHLORIDE | IMIPRAMINE P...)
Affinity DataEC50:  1.00E+4nMAssay Description:Half maximal inhibition of Prion protein PrPsc formation was assayed in ScN2a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed