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Found 15 of ic50 for UniProtKB: Q9QUR6
TargetProlyl endopeptidase(Mus musculus)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50155838((S)-1-((S)-1-(4-phenylbutanoyl)pyrrolidine-2-carbo...)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of PREP in C57BL/6 mouse cortex homogenate assessed as formation of 7-amido-4-methylcoumarin using Suc-Gly-Pro-amido-4-methylcoumarin as s...More data for this Ligand-Target Pair
TargetProlyl endopeptidase(Mus musculus)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50005870(CHEMBL3236271)
Affinity DataIC50:  3.10nMAssay Description:Competitive inhibition of mouse brain prolyl oligopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Mus musculus)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50529486(CHEMBL4549821)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of PREP in C57BL/6 mouse cortex homogenate assessed as formation of 7-amido-4-methylcoumarin using Suc-Gly-Pro-amido-4-methylcoumarin as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Mus musculus)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50051539((S)-4-phenyl-1-(2-(pyrrolidine-1-carbonyl)pyrrolid...)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of mouse brain POPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Mus musculus)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50529474(CHEMBL4528594)
Affinity DataIC50:  91nMAssay Description:Inhibition of PREP in C57BL/6 mouse cortex homogenate assessed as formation of 7-amido-4-methylcoumarin using Suc-Gly-Pro-amido-4-methylcoumarin as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Mus musculus)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50529487(CHEMBL4465322)
Affinity DataIC50:  264nMAssay Description:Inhibition of PREP in C57BL/6 mouse cortex homogenate assessed as formation of 7-amido-4-methylcoumarin using Suc-Gly-Pro-amido-4-methylcoumarin as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Mus musculus)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50529483(CHEMBL4556841)
Affinity DataIC50:  298nMAssay Description:Inhibition of PREP in C57BL/6 mouse cortex homogenate assessed as formation of 7-amido-4-methylcoumarin using Suc-Gly-Pro-amido-4-methylcoumarin as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Mus musculus)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50529494(CHEMBL4540171)
Affinity DataIC50:  5.14E+3nMAssay Description:Inhibition of PREP in C57BL/6 mouse cortex homogenate assessed as formation of 7-amido-4-methylcoumarin using Suc-Gly-Pro-amido-4-methylcoumarin as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Mus musculus)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50529475(CHEMBL4588059)
Affinity DataIC50:  6.21E+3nMAssay Description:Inhibition of PREP in C57BL/6 mouse cortex homogenate assessed as formation of 7-amido-4-methylcoumarin using Suc-Gly-Pro-amido-4-methylcoumarin as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Mus musculus)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50529484(CHEMBL4586782)
Affinity DataIC50:  1.21E+4nMAssay Description:Inhibition of PREP in C57BL/6 mouse cortex homogenate assessed as formation of 7-amido-4-methylcoumarin using Suc-Gly-Pro-amido-4-methylcoumarin as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Mus musculus)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50529491(CHEMBL4520738)
Affinity DataIC50:  1.35E+4nMAssay Description:Inhibition of PREP in C57BL/6 mouse cortex homogenate assessed as formation of 7-amido-4-methylcoumarin using Suc-Gly-Pro-amido-4-methylcoumarin as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Mus musculus)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50529485(CHEMBL4475037)
Affinity DataIC50:  2.88E+4nMAssay Description:Inhibition of PREP in C57BL/6 mouse cortex homogenate assessed as formation of 7-amido-4-methylcoumarin using Suc-Gly-Pro-amido-4-methylcoumarin as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Mus musculus)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50529489(CHEMBL4551013)
Affinity DataIC50:  3.52E+4nMAssay Description:Inhibition of PREP in C57BL/6 mouse cortex homogenate assessed as formation of 7-amido-4-methylcoumarin using Suc-Gly-Pro-amido-4-methylcoumarin as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Mus musculus)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50529495(CHEMBL4441906)
Affinity DataIC50:  1.54E+5nMAssay Description:Inhibition of PREP in C57BL/6 mouse cortex homogenate assessed as formation of 7-amido-4-methylcoumarin using Suc-Gly-Pro-amido-4-methylcoumarin as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Mus musculus)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50529490(CHEMBL4436952)
Affinity DataIC50:  4.57E+5nMAssay Description:Inhibition of PREP in C57BL/6 mouse cortex homogenate assessed as formation of 7-amido-4-methylcoumarin using Suc-Gly-Pro-amido-4-methylcoumarin as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed