Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 130nMAssay Description:Induction of degradation of endogenous HMGCR in CHO-7 cells assessed as decrease in protein level incubated for 16 hrs in sterol-depleted medium by i...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 220nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 280nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 390nMAssay Description:Induction of HMGCR degradation in CHO-7 cells incubated for 16 hrs by immunoblotting assayMore data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 410nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 410nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 410nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 410nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 410nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 410nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 430nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 430nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 430nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 480nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 520nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 530nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 630nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 650nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 730nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 760nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 820nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 830nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 980nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 1.09E+3nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 1.26E+3nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 1.63E+3nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 1.84E+3nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 2.03E+3nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 2.66E+3nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 2.73E+3nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 3.37E+3nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 3.99E+3nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 4.47E+3nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 4.80E+3nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 4.94E+3nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 5.02E+3nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 5.41E+3nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 5.81E+3nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 8.16E+3nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 8.25E+3nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 8.80E+3nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 1.26E+4nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 2.81E+4nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 3.14E+4nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Cricetulus griseus)
East China Normal University
Curated by ChEMBL
East China Normal University
Curated by ChEMBL
Affinity DataEC50: 4.39E+4nMAssay Description:Induction of degradation of hamster HMGCR (TM1-8)-GFP (1 to 346 residues) transfected in CHO-7 cells incubated for 16 hrs in sterol-depleted medium b...More data for this Ligand-Target Pair