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Found 25 of ic50 for UniProtKB: P23919
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50550238(CHEMBL4749381)
Affinity DataIC50:  350nMAssay Description:Inhibition of GST-tagged human TMPK expressed in Escherichia coli BL21 incubated for 10 mins by luciferase-coupled TMPK assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50550239(CHEMBL4758532)
Affinity DataIC50:  470nMAssay Description:Inhibition of GST-tagged human TMPK expressed in Escherichia coli BL21 incubated for 10 mins by luciferase-coupled TMPK assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50365395(CHEMBL395814)
Affinity DataIC50:  1.53E+3nMAssay Description:Inhibition of human thymidylate kinase using dTMP as substrate after 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50550240(CHEMBL4757635)
Affinity DataIC50:  1.65E+3nMAssay Description:Inhibition of GST-tagged human TMPK expressed in Escherichia coli BL21 incubated for 10 mins by luciferase-coupled TMPK assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50367702(CHEMBL606084)
Affinity DataIC50:  4.00E+3nMAssay Description:Concentration required to reduce Thymidylate kinase rate by 50% in human blast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50367696(CHEMBL605435)
Affinity DataIC50:  6.00E+3nMAssay Description:Concentration required to reduce Thymidylate kinase rate by 50% in human blast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50367698(CHEMBL604405)
Affinity DataIC50:  6.00E+3nMAssay Description:Concentration required to reduce Thymidylate kinase rate by 50% in human blast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50366828(CHEMBL1236157)
Affinity DataIC50:  8.00E+3nMAssay Description:Concentration required to reduce Thymidylate kinase rate by 50% in human blast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50398957(CHEMBL2179281)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of human thymidylate kinase assessed as effect on ATP production by Escherichia coli DdlA and Malachite green reagent based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50398958(CHEMBL2179279)
Affinity DataIC50:  4.34E+4nMAssay Description:Inhibition of human thymidylate kinase assessed as effect on ATP production by Escherichia coli DdlA and Malachite green reagent based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50398959(CHEMBL2179277)
Affinity DataIC50:  6.20E+4nMAssay Description:Inhibition of human thymidylate kinase assessed as effect on ATP production by Escherichia coli DdlA and Malachite green reagent based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50365393(CHEMBL1956669)
Affinity DataIC50:  1.23E+5nMAssay Description:Inhibition of human thymidylate kinase using dTMP as substrate after 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50365394(CHEMBL1956676)
Affinity DataIC50:  1.24E+5nMAssay Description:Inhibition of human thymidylate kinase using dTMP as substrate after 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50398961(CHEMBL2179269)
Affinity DataIC50:  1.50E+5nMAssay Description:Inhibition of human thymidylate kinase assessed as effect on ATP production by Escherichia coli DdlA and Malachite green reagent based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50398960(CHEMBL2179273)
Affinity DataIC50:  1.50E+5nMAssay Description:Inhibition of human thymidylate kinase assessed as effect on ATP production by Escherichia coli DdlA and Malachite green reagent based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50428613(CHEMBL2331747)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human thymidylate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50398962(CHEMBL2179669)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human thymidylate kinase assessed as effect on ATP production by Escherichia coli DdlA and Malachite green reagent based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50365391(CHEMBL1956642)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human thymidylate kinase using dTMP as substrate after 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50365390(CHEMBL1956634)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human thymidylate kinase using dTMP as substrate after 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50365392(CHEMBL1956668)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human thymidylate kinase using dTMP as substrate after 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50367703(CHEMBL1794614 | CHEMBL603793)
Affinity DataIC50:  2.90E+5nMAssay Description:Concentration required to reduce Thymidylate kinase rate by 50% in human blast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50367697(CHEMBL606301)
Affinity DataIC50:  3.40E+5nMAssay Description:Concentration required to reduce Thymidylate kinase rate by 50% in human blast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50367704(CHEMBL604419)
Affinity DataIC50:  7.30E+5nMAssay Description:Concentration required to reduce Thymidylate kinase rate by 50% in human blast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50367699(CHEMBL604420)
Affinity DataIC50: >1.00E+6nMAssay Description:Concentration required to reduce Thymidylate kinase rate by 50% in human blast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50367701(CHEMBL605228)
Affinity DataIC50:  1.23E+6nMAssay Description:Concentration required to reduce Thymidylate kinase rate by 50% in human blast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed