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Found 17 of ic50 for UniProtKB: P97772
TargetMetabotropic glutamate receptor 1(Mus musculus)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50333367(6-(1-(2-fluoropyridin-3-yl)-5-methyl-1H-1,2,3-tria...)
Affinity DataIC50:  1.40nMAssay Description:Binding affinity to mouse mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Mus musculus)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50273899(CHEMBL456823 | tert-Butyl-4-[1-(2-fuluoropyridine-...)
Affinity DataIC50:  1.5nMAssay Description:Antagonist activity at mouse mGluR1 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Mus musculus)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50273942(4-(1-(2-fluoropyridin-3-yl)-5-methyl-1H-1,2,3-tria...)
Affinity DataIC50:  3.10nMAssay Description:Antagonist activity at mouse mGluR1 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Mus musculus)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50273941(CHEMBL456196 | iso-Propyl-4-[1-(2-fuluoropyridine-...)
Affinity DataIC50:  3.30nMAssay Description:Antagonist activity at mouse mGluR1 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Mus musculus)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50273898(CHEMBL452618 | tert-Butyl-4-[1-(2-fuluoropyridine-...)
Affinity DataIC50:  12nMAssay Description:Antagonist activity at mouse mGluR1 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Mus musculus)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50273829(CHEMBL461673 | tert-Butyl-4-[1-(2-fluorophenyl)-1H...)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at mouse mGluR1 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Mus musculus)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50273828(CHEMBL511355 | tert-Butyl-4-(1-phenyl-1H-1,2,3-tri...)
Affinity DataIC50:  24nMAssay Description:Antagonist activity at mouse mGluR1 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Mus musculus)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50273863(CHEMBL460827 | tert-Butyl-4-[1-(4-fuluorophenyl)-1...)
Affinity DataIC50:  31nMAssay Description:Antagonist activity at mouse mGluR1 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Mus musculus)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50273830(CHEMBL460391 | tert-Butyl-4-[1-(3-fuluorophenyl)-1...)
Affinity DataIC50:  39nMAssay Description:Antagonist activity at mouse mGluR1 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Mus musculus)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50273864(CHEMBL511352 | tert-Butyl-4-[1-(2-methylphenyl)-1H...)
Affinity DataIC50:  58nMAssay Description:Antagonist activity at mouse mGluR1 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Mus musculus)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50273895(CHEMBL457872 | tert-Butyl-4-[1-pyridin-2-yl-1H-1,2...)
Affinity DataIC50:  150nMAssay Description:Antagonist activity at mouse mGluR1 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Mus musculus)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50273867(1-(3,3-Dimethylbutanolyl)-4-[1-(2-fluorophenyl)-1H...)
Affinity DataIC50:  160nMAssay Description:Antagonist activity at mouse mGluR1 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Mus musculus)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50273896(CHEMBL453249 | tert-Butyl-4-[1-pyridin-3-yl-1 H-1,...)
Affinity DataIC50:  180nMAssay Description:Antagonist activity at mouse mGluR1 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Mus musculus)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50273940(CHEMBL457026 | iso-Propyl-4-[1-(2-fuluoropyridine-...)
Affinity DataIC50:  180nMAssay Description:Antagonist activity at mouse mGluR1 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Mus musculus)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50273866(CHEMBL461034 | N-(tert-Butyl)-4-[1-(2-fluorophenyl...)
Affinity DataIC50:  290nMAssay Description:Antagonist activity at mouse mGluR1 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Mus musculus)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50273897(CHEMBL457873 | tert-Butyl-4-[1-pyridin-4-yl-1 H-1,...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at mouse mGluR1 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Mus musculus)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50273865(CHEMBL461033 | tert-Butyl-4-[1-(2-methoxylphenyl)-...)
Affinity DataIC50:  1.60E+3nMAssay Description:Antagonist activity at mouse mGluR1 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed