Compile Data Set for Download or QSAR
maximum 50k data
Found 9 of ec50 for UniProtKB: Q8CFK4
TargetTyrosine-protein kinase(Mus musculus)
The University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154582(6-[1,3]Dioxan-2-yl-quinolin-2-ylamine | CHEMBL4266...)
Affinity DataEC50:  2.60E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase(Mus musculus)
The University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154587(6-[1,3]Dioxolan-2-yl-quinolin-2-ylamine | CHEMBL36...)
Affinity DataEC50:  3.40E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase(Mus musculus)
The University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154591(6-Bromo-quinolin-2-ylamine | CHEMBL189197)
Affinity DataEC50:  5.80E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase(Mus musculus)
The University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154590(6-Methoxy-quinolin-2-ylamine | CHEMBL188730)
Affinity DataEC50:  6.30E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase(Mus musculus)
The University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154583(6-Methyl-quinolin-2-ylamine | CHEMBL361660)
Affinity DataEC50:  7.50E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase(Mus musculus)
The University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154589(6-Chloro-quinolin-2-ylamine | CHEMBL189514)
Affinity DataEC50:  7.60E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase(Mus musculus)
The University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154584(6-Fluoro-quinolin-2-ylamine | CHEMBL185917)
Affinity DataEC50:  1.50E+5nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase(Mus musculus)
The University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM14322(2-Aminoquinoline 1 | 2-aminoquinoline | CHEMBL6123...)
Affinity DataEC50:  1.60E+5nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase(Mus musculus)
The University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154588(5,6,7,8-Tetrahydro-quinolin-2-ylamine | CHEMBL1888...)
Affinity DataEC50:  2.15E+5nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed