Compile Data Set for Download or QSAR
maximum 50k data
Found 9 of kd for UniProtKB: Q8CFK4
TargetTyrosine-protein kinase(Mus musculus)
The University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154586(6-(5,5-Dimethyl-[1,3]dioxan-2-yl)-quinolin-2-ylami...)
Affinity DataKd:  2.20E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase(Mus musculus)
The University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154587(6-[1,3]Dioxolan-2-yl-quinolin-2-ylamine | CHEMBL36...)
Affinity DataKd:  4.00E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase(Mus musculus)
The University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154582(6-[1,3]Dioxan-2-yl-quinolin-2-ylamine | CHEMBL4266...)
Affinity DataKd:  5.20E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase(Mus musculus)
The University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154583(6-Methyl-quinolin-2-ylamine | CHEMBL361660)
Affinity DataKd:  6.10E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase(Mus musculus)
The University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM14322(2-Aminoquinoline 1 | 2-aminoquinoline | CHEMBL6123...)
Affinity DataKd:  1.25E+5nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase(Mus musculus)
The University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50084506(CHEMBL319543 | Methyl-quinolin-2-yl-amine)
Affinity DataKd:  3.80E+5nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase(Mus musculus)
The University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM14320(1-amino-isoquinoline | CHEMBL62083 | Fragment 17 |...)
Affinity DataKd:  6.50E+5nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase(Mus musculus)
The University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154585(CHEMBL187951 | Quinazolin-2-ylamine)
Affinity DataKd:  8.00E+5nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase(Mus musculus)
The University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50013712(2-aminopyridin | 2-aminopyridine | CHEMBL21619 | P...)
Affinity DataKd: >4.00E+6nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed