Compile Data Set for Download or QSAR
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Found 13 of ec50 for UniProtKB: Q9EP66
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50384640(CHEMBL2036954)
Affinity DataEC50:  4nMAssay Description:Agonist activity at mouse GPR109aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50337038(5-(3-cyclopropylpropyl)-2-(difluoromethyl)-3H-pyra...)
Affinity DataEC50:  4nMAssay Description:Agonist activity at mouse GPR109aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50384637(CHEMBL2036951)
Affinity DataEC50:  5nMAssay Description:Agonist activity at mouse GPR109aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50384612(CHEMBL2036958)
Affinity DataEC50:  6nMAssay Description:Agonist activity at mouse GPR109aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50384616(CHEMBL2036813)
Affinity DataEC50:  12nMAssay Description:Agonist activity at mouse GPR109aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50337024(2-(difluoromethyl)-5-(3-(1-methylcyclopropyl)propy...)
Affinity DataEC50:  15nMAssay Description:Agonist activity at mouse GPR109aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM23515(CHEMBL573 | Niacin | Nicotinic Acid | [5, 6-3H]-ni...)
Affinity DataEC50:  29nMAssay Description:Agonist activity at mouse GPR109aMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM23515(CHEMBL573 | Niacin | Nicotinic Acid | [5, 6-3H]-ni...)
Affinity DataEC50:  29nMAssay Description:Agonist activity at mouse GPR109aMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50313976(2-({3-[3-(5-hydroxypyridin-2-yl)-1,2,4-oxadiazol-5...)
Affinity DataEC50:  240nMAssay Description:Agonist activity at mouse GPR109A receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50273099(3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocyclopenta[...)
Affinity DataEC50:  400nMAssay Description:Agonist activity against mouse GPR109a assessed as GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50132140(1,4,5,6-Tetrahydro-cyclopentapyrazole-3-carboxylic...)
Affinity DataEC50:  500nMAssay Description:Agonist activity against mouse GPR109a assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50273099(3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocyclopenta[...)
Affinity DataEC50:  1.08E+3nMAssay Description:Agonist activity against mouse GPR109a assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50216525(6-Methyl-1,4,5,6-tetrahydrocyclopenta[c]pyrazole-3...)
Affinity DataEC50:  1.22E+4nMAssay Description:Agonist activity against mouse GPR109a assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed