Compile Data Set for Download or QSAR
maximum 50k data
Found 76 of ic50 for UniProtKB: P51683
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50331722(CHEMBL1290636 | N-(2-((3S,4S)-4-ethoxy-1-(cis-4-ph...)
Affinity DataIC50:  1.90nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 after 30 mins by gamma counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50331723(CHEMBL1290637 | N-(2-oxo-2-((3S,4S)-1-(cis-4-pheny...)
Affinity DataIC50:  1.90nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 after 30 mins by gamma counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50331727(CHEMBL1289203 | N-(2-((3S,4S)-4-ethoxy-1-(cis-4-hy...)
Affinity DataIC50:  2.10nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 after 30 mins by gamma counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50337619(((1S,3R)-1-isopropyl-3-((3S,4S)-3-methoxytetrahydr...)
Affinity DataIC50:  2.80nMAssay Description:Binding affinity to mouse CCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212146(1-ethyl-N-{[3-fluoro-5-(trifluoromethyl)phenyl]met...)
Affinity DataIC50:  3.5nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50381177(CHEMBL2018386)
Affinity DataIC50:  4nMAssay Description:Antagonist activity at CCR2 in mouse monocytes assessed as inhibition of MCP1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212136((1S,3R)-N-{[3-fluoro-5-(trifluoromethyl)phenyl]met...)
Affinity DataIC50:  5nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212128((1R,3R)-N-{[3-fluoro-5-(trifluoromethyl)phenyl]met...)
Affinity DataIC50:  7.5nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50331728(CHEMBL1289316 | N-(2-((3S,4S)-1-(cis-4-(benzo[d][1...)
Affinity DataIC50:  7.80nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 after 30 mins by gamma counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212127((1S,3R)-1-cyclopropyl-N-{[3-fluoro-5-(trifluoromet...)
Affinity DataIC50:  8nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50331728(CHEMBL1289316 | N-(2-((3S,4S)-1-(cis-4-(benzo[d][1...)
Affinity DataIC50:  9.5nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 after 30 mins by gamma counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50331726(CHEMBL1289083 | N-(2-((3S,4S)-4-ethoxy-1-(cis-4-hy...)
Affinity DataIC50:  10nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 after 30 mins by gamma counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50331727(CHEMBL1289203 | N-(2-((3S,4S)-4-ethoxy-1-(cis-4-hy...)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at mouse CCR2 assessed as inhibition of MCP1 induced chemotaxis after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50331722(CHEMBL1290636 | N-(2-((3S,4S)-4-ethoxy-1-(cis-4-ph...)
Affinity DataIC50:  14nMAssay Description:Antagonist activity at mouse CCR2 assessed as inhibition of MCP1 induced chemotaxis after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212145((1S,3R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}...)
Affinity DataIC50:  15nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212131(1-(cyclopropylmethyl)-N-{[3-fluoro-5-(trifluoromet...)
Affinity DataIC50:  15nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50382932(CHEMBL2029422)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at mouse CCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212122((1R,3R)-N-{[3-fluoro-5-(trifluoromethyl)phenyl]met...)
Affinity DataIC50:  17nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212134(CHEMBL231038 | N-{[3-fluoro-5-(trifluoromethyl)phe...)
Affinity DataIC50:  17nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50382932(CHEMBL2029422)
Affinity DataIC50:  17nMAssay Description:Binding affinity to mouse CCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212126(CHEMBL388007 | N-{[3,5-bis(trifluoromethyl)phenyl]...)
Affinity DataIC50:  17.5nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50363942(CHEMBL1951766)
Affinity DataIC50:  18nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 after 30 mins by gamma counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212139((1R,3R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}...)
Affinity DataIC50:  26nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212138((1S,3R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}...)
Affinity DataIC50:  44.3nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212135(CHEMBL266017 | N-{[3,5-bis(trifluoromethyl)phenyl]...)
Affinity DataIC50:  45nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50578294(Bms 813160 | Bms-813160)
Affinity DataIC50:  45nMAssay Description:Displacement of [125I]-CCL2 from mouse CCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50331725(CHEMBL1288324 | N-(2-((3S,4S)-4-(benzyloxy)-1-(cis...)
Affinity DataIC50:  51nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 after 30 mins by gamma counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50331724(CHEMBL1290754 | N-(2-((3S,4S)-4-butoxy-1-(cis-4-ph...)
Affinity DataIC50:  54nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 after 30 mins by gamma counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212140((1S,3R)-N-{[3-fluoro-5-(trifluoromethyl)phenyl]met...)
Affinity DataIC50:  57nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212142(CHEMBL230078 | N-{[3,5-bis(trifluoromethyl)phenyl]...)
Affinity DataIC50:  63.5nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212124((1R,3R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}...)
Affinity DataIC50:  64nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212130((1R,3R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}...)
Affinity DataIC50:  65.5nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212125(CHEMBL389610 | N-{[3-fluoro-5-(trifluoromethyl)phe...)
Affinity DataIC50:  74nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50198119(CHEMBL231340 | N-{[3,5-bis(trifluoromethyl)phenyl]...)
Affinity DataIC50:  79nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 expressed in monocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50198134(CHEMBL395289 | N-{[3,5-bis(trifluoromethyl)phenyl]...)
Affinity DataIC50:  81nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 expressed in monocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212144(CHEMBL230831 | N-{[3,5-bis(trifluoromethyl)phenyl]...)
Affinity DataIC50:  93nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50198139(CHEMBL397717 | N-{4-[1-({[3,5-bis(trifluoromethyl)...)
Affinity DataIC50:  111nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 expressed in monocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212141((1S,3R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}...)
Affinity DataIC50:  126nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212123(CHEMBL231143 | N-{[3-fluoro-5-(trifluoromethyl)phe...)
Affinity DataIC50:  128nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50211499((1S,3R)-N-[3,5-bis(trifluoromethyl)benzyl]-1-methy...)
Affinity DataIC50:  130nMAssay Description:Displacement of [125]hMCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212129(1-(cyclobutylmethyl)-N-{[3-fluoro-5-(trifluorometh...)
Affinity DataIC50:  147nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50363942(CHEMBL1951766)
Affinity DataIC50:  156nMAssay Description:Antagonist activity at mouse CCR2 assessed as inhibition of MCP1-induced chemotaxis after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50331723(CHEMBL1290637 | N-(2-oxo-2-((3S,4S)-1-(cis-4-pheny...)
Affinity DataIC50:  158nMAssay Description:Antagonist activity at mouse CCR2 assessed as inhibition of MCP1 induced chemotaxis after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50198116(CHEMBL438128 | N-{[3,5-bis(trifluoromethyl)phenyl]...)
Affinity DataIC50:  165nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 expressed in monocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50198111(CHEMBL231149 | N-{4-[1-({[3,5-bis(trifluoromethyl)...)
Affinity DataIC50:  186nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 expressed in monocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50331715(CHEMBL1290412 | N-(2-((3S,4S)-4-hydroxy-1-(cis-4-p...)
Affinity DataIC50:  186nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 after 30 mins by gamma counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212143((1R,3R)-N-{[3-fluoro-5-(trifluoromethyl)phenyl]met...)
Affinity DataIC50:  193nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50331715(CHEMBL1290412 | N-(2-((3S,4S)-4-hydroxy-1-(cis-4-p...)
Affinity DataIC50:  265nMAssay Description:Antagonist activity at mouse CCR2 assessed as inhibition of MCP1 induced chemotaxis after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212133(CHEMBL398001 | N-{[3,5-bis(trifluoromethyl)phenyl]...)
Affinity DataIC50:  279nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte

Curated by ChEMBL
LigandPNGBDBM50212137((1R,3R)-N-{[3,5-bis(trifluoromethyl)phenyl]methyl}...)
Affinity DataIC50:  351nMAssay Description:Displacement of [125I]MCP1 from mouse CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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