Affinity DataKi: 300nMAssay Description:In vitro inhibitory activity against Catechol-O-methyltransferase from porcine liver; Competitive mode of inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:In vitro inhibitory activity against Catechol-O-methyltransferase from porcine liver; Competitive mode of inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 6.60E+3nMAssay Description:In vitro inhibitory activity against Catechol-O-methyltransferase from porcine liver; Uncompetitive mode of inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 1.35E+4nMAssay Description:Compound was evaluated for reversible inhibition of Catechol O-methyltransferase with variable AdoMet and saturating catechol as substrate (mixed inh...More data for this Ligand-Target Pair
Affinity DataKi: 1.72E+4nMAssay Description:Compound was evaluated for reversible inhibition of Catechol O-methyltransferase with saturating AdoMet and variable catechol as substrate (noncompet...More data for this Ligand-Target Pair
Affinity DataKi: 2.67E+4nMAssay Description:In vitro inhibitory activity against Catechol-O-methyltransferase from porcine liver; Uncompetitive mode of inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 3.50E+4nMAssay Description:In vitro inhibitory activity against Catechol-O-methyltransferase from porcine liver; Uncompetitive mode of inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 1.36E+5nMAssay Description:In vitro inhibitory activity against Catechol-O-methyltransferase from porcine liver; Uncompetitive mode of inhibitionMore data for this Ligand-Target Pair