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Found 30 of ic50 for UniProtKB: Q9Y2T5
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556715(CHEMBL4782344)
Affinity DataIC50:  630nMAssay Description:In vitro inhibitory activity against beta-2 adrenergic receptor was measured by the inhibition of isoproterenol-induced relaxation of PGF2-alpha cont...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556717(CHEMBL4780703)
Affinity DataIC50:  630nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556698(CHEMBL2375494)
Affinity DataIC50:  650nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556698(CHEMBL2375494)
Affinity DataIC50:  650nMAssay Description:In vitro inhibitory activity against beta-2 adrenergic receptor was measured by the inhibition of isoproterenol-induced relaxation of PGF2-alpha cont...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556715(CHEMBL4782344)
Affinity DataIC50:  880nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556716(CHEMBL4796964)
Affinity DataIC50:  910nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556721(CHEMBL4790746)
Affinity DataIC50:  1.01E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556719(CHEMBL4782590)
Affinity DataIC50:  1.08E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556710(CHEMBL4741257)
Affinity DataIC50:  1.23E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556706(CHEMBL4797370)
Affinity DataIC50:  1.49E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556718(CHEMBL4787771)
Affinity DataIC50:  1.52E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556699(CHEMBL4746541)
Affinity DataIC50:  1.64E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556705(CHEMBL4793323)
Affinity DataIC50:  1.72E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556708(CHEMBL4795327)
Affinity DataIC50:  1.76E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556700(CHEMBL4761208)
Affinity DataIC50:  1.81E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556722(CHEMBL4791780)
Affinity DataIC50:  1.81E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556720(CHEMBL4745132)
Affinity DataIC50:  1.82E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556709(CHEMBL4783011)
Affinity DataIC50:  2.37E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556703(CHEMBL4761078)
Affinity DataIC50:  2.57E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556701(CHEMBL4746014)
Affinity DataIC50:  2.63E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556702(CHEMBL4763588)
Affinity DataIC50:  2.82E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556704(CHEMBL4740701)
Affinity DataIC50:  3.02E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556713(CHEMBL4748854)
Affinity DataIC50:  3.29E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556714(CHEMBL4777734)
Affinity DataIC50:  3.54E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556707(CHEMBL4762863)
Affinity DataIC50:  3.87E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556723(CHEMBL240484)
Affinity DataIC50:  5.45E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556723(CHEMBL240484)
Affinity DataIC50:  5.45E+3nMAssay Description:In vitro inhibitory activity against beta-2 adrenergic receptor was measured by the inhibition of isoproterenol-induced relaxation of PGF2-alpha cont...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556712(CHEMBL4798117)
Affinity DataIC50:  7.64E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556711(CHEMBL4755423)
Affinity DataIC50:  8.13E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50405604(CHEMBL5279049)
Affinity DataIC50:  1.20E+4nMAssay Description:In vitro inhibitory activity against beta-2 adrenergic receptor was measured by the inhibition of isoproterenol-induced relaxation of PGF2-alpha cont...More data for this Ligand-Target Pair
In DepthDetails PubMed