TargetMuscarinic acetylcholine receptor M5(Mus musculus)
Johns Hopkins Medical Institutions
Curated by ChEMBL
Johns Hopkins Medical Institutions
Curated by ChEMBL
Affinity DataIC50: 3.30nMAssay Description:Ability (10 ug/kg) to inhibit binding of [125I]iododexetimide to muscarinic receptor in miceMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(Mus musculus)
Johns Hopkins Medical Institutions
Curated by ChEMBL
Johns Hopkins Medical Institutions
Curated by ChEMBL
Affinity DataIC50: 750nMAssay Description:Ability (10 ug/kg) to inhibit binding of [125I]iododexetimide to muscarinic receptor in miceMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(Mus musculus)
Johns Hopkins Medical Institutions
Curated by ChEMBL
Johns Hopkins Medical Institutions
Curated by ChEMBL
Affinity DataIC50: 8.90E+3nMAssay Description:Ability (10 ug/kg) to inhibit binding of [125I]iododexetimide to muscarinic receptor in miceMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Mus musculus)
Sri International
Curated by ChEMBL
Sri International
Curated by ChEMBL
Affinity DataIC50: 2.20E+4nMAssay Description:Compound was tested for the binding affinity towards muscarinic receptor in mouse brain membraneMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Mus musculus)
Sri International
Curated by ChEMBL
Sri International
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Compound was tested for the binding affinity towards muscarinic receptor in mouse brain membraneMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Mus musculus)
Sri International
Curated by ChEMBL
Sri International
Curated by ChEMBL
Affinity DataIC50: 8.00E+4nMAssay Description:Compound was tested for the binding affinity towards muscarinic acetylcholine receptor in mouse brain membraneMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Mus musculus)
Sri International
Curated by ChEMBL
Sri International
Curated by ChEMBL
Affinity DataIC50: 1.60E+5nMAssay Description:Compound was tested for the competitive inhibition of phosphonylation of Eel acetylcholinesterase (AChE)More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Mus musculus)
Sri International
Curated by ChEMBL
Sri International
Curated by ChEMBL
Affinity DataIC50: 1.70E+5nMAssay Description:Compound was tested for the binding affinity towards muscarinic receptor in mouse brain membraneMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Mus musculus)
Sri International
Curated by ChEMBL
Sri International
Curated by ChEMBL
Affinity DataIC50: 1.00E+6nMAssay Description:Compound was tested for the competitive inhibition of phosphonylation of Eel acetylcholinesterase (AChE)More data for this Ligand-Target Pair