Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ic50 for UniProtKB: Q920H4
TargetMuscarinic acetylcholine receptor M5(Mus musculus)
Johns Hopkins Medical Institutions

Curated by ChEMBL
LigandPNGBDBM50228206(Dexetimide | R-16470 [as hydrochloride])
Affinity DataIC50:  3.30nMAssay Description:Ability (10 ug/kg) to inhibit binding of [125I]iododexetimide to muscarinic receptor in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Mus musculus)
Johns Hopkins Medical Institutions

Curated by ChEMBL
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataIC50:  750nMAssay Description:Ability (10 ug/kg) to inhibit binding of [125I]iododexetimide to muscarinic receptor in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Mus musculus)
Johns Hopkins Medical Institutions

Curated by ChEMBL
LigandPNGBDBM50018556((+)-1'-benzyl-3-phenyl-3,4'-bipiperidine-2,6-dione...)
Affinity DataIC50:  8.90E+3nMAssay Description:Ability (10 ug/kg) to inhibit binding of [125I]iododexetimide to muscarinic receptor in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed