Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
Ligand InfoPDB
Affinity DataKi: 0.140nM ΔG°: -13.1kcal/molepH: 7.4 T: 2°CAssay Description:[3H]PDBu binding to the C1 domains of MRCK alpha/beta and PKC alpha/delta was measured using the polyethylene glycol precipitation assay.More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Displacement of [3H]PDBu from PKCdelta C1B domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:Inhibition of [3H]PDBu binding to PKC delta C1B peptideMore data for this Ligand-Target Pair
Affinity DataKi: 0.440nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCdelta expressed in Sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Displacement of [3H]PDBu from PKCdelta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Displacement of 3[H]PDBu from Protein kinase C delta C1a domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding affinity for human recombinant protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding affinity for human recombinant protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inhibition of [3H]-phorbol 12,13-dibutyrate (PDBu) binding to human recombinant protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding affinity for human recombinant protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]- PDBu from recombinant PKC delta expressed in baculovirusMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inhibition of [3H]-PDBu binding to PKC delta wild typeMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Inhibition of [3H]PDBu binding to C1b domain of protein kinase C delta with phosphatidylserineMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity for isolated C1b domain of protein kinase C-deltaMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of 3[H]PDBu from Protein kinase C delta C1a domainMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of [3H]PDBu binding to recombinant full length human PKCdelta expressed in baculovirus expression system incubated for 5 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 1.16nM ΔG°: -11.9kcal/molepH: 7.4 T: 2°CAssay Description:[3H]PDBu binding to the C1 domains of MRCK alpha/beta and PKC alpha/delta was measured using the polyethylene glycol precipitation assay.More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of [3H]-PDBu binding to C1b domain of protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity for isolated C1b domain of protein kinase C-deltaMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of [3H]PDBu binding to recombinant full length human PKCdelta expressed in baculovirus expression system incubated for 5 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta-C1B domain peptide (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity to PKCdeltaC1b in presence of phospholipidMore data for this Ligand-Target Pair
Affinity DataKi: 1.54nM ΔG°: -11.7kcal/molepH: 7.4 T: 2°CAssay Description:[3H]PDBu binding to the C1 domains of MRCK alpha/beta and PKC alpha/delta was measured using the polyethylene glycol precipitation assay.More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Inhibition of [3H]PDBu binding to recombinant full length human PKCdelta expressed in baculovirus expression system incubated for 5 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Inhibition of human Protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]-PDBu from protein kinase C delta C1b domainMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Inhibition of [3H]PDBu binding to recombinant full length human PKCdelta expressed in baculovirus expression system incubated for 5 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Displacement of [3H]PDBu form human PKCdelta in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Inhibition of [3H]PDBu binding to recombinant full length human PKCdelta expressed in baculovirus expression system incubated for 5 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Inhibition of [3H]PDBu binding to C1b domain of protein kinase C delta with phosphatidylserineMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Inhibition of [3H]PDBu binding to recombinant full length human PKCdelta expressed in baculovirus expression system incubated for 5 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Inhibition of [3H]PDBu binding to recombinant full length human PKCdelta expressed in baculovirus expression system incubated for 5 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta-C1B domain peptide (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Inhibition of [3H]PDBu binding to recombinant full length human PKCdelta expressed in baculovirus expression system incubated for 5 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition of [3H]PDBu binding to recombinant full length human PKCdelta expressed in baculovirus expression system incubated for 5 mins by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta-C1B domain peptide (unknown origin)More data for this Ligand-Target Pair