Compile Data Set for Download or QSAR
Report error Found 8 of kd for UniProtKB: Q8NER1
TargetTransient receptor potential cation channel subfamily V member 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50241484BDBM50241484(CHEMBL4095861)
Affinity DataKd:  0.589nMAssay Description:Binding affinity to human TRPV1 expressed in CHO cells after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50241484BDBM50241484(CHEMBL4095861)
Affinity DataKd:  0.590nMAssay Description:Binding affinity to human TRPV1 expressed in CHO cells after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50241485BDBM50241485(CHEMBL4060041)
Affinity DataKd:  1.20nMAssay Description:Binding affinity to human TRPV1 expressed in CHO cells after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 20458BDBM20458(A-778317 | 1-[(1R)-5-tert-butyl-2,3-dihydro-1H-ind...)
Affinity DataKd:  3.40nMAssay Description:Displacement of [3H]A-778317 from human TRPV1 expressed in CHO cell membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50329104BDBM50329104(Indole alkaloid derivative | voacangine | CHEMBL18...)
Affinity DataKd:  2.00E+4nMAssay Description:Competitive antagonist activity at human brain TRPV1 expressed in HEK293T cells assessed as inhibition of CAP-induced intracellular Ca2+ influx prein...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50618693BDBM50618693(CHEMBL5420817)
Affinity DataKd:  4.03E+4nMAssay Description:Binding affinity to human TRPV1 assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50318484BDBM50318484(CHEMBL190461 | 2-((1R,6R)-6-Isopropenyl-3-methyl-c...)
Affinity DataKd:  1.10E+5nMAssay Description:Binding affinity to human TRPV1 assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50618694BDBM50618694(CHEMBL5430046)
Affinity DataKd:  2.73E+5nMAssay Description:Binding affinity to human TRPV1 assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed