Compile Data Set for Download or QSAR
maximum 50k data
Found 35 of ic50 for UniProtKB: Q9JIM1
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457379(CHEMBL4211925)
Affinity DataIC50:  14nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457390(CHEMBL4208680)
Affinity DataIC50:  17nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457381(CHEMBL4211194)
Affinity DataIC50:  18nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457387(CHEMBL4215413)
Affinity DataIC50:  24nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457386(CHEMBL4212967)
Affinity DataIC50:  26nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409054(3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-1-(5-(meth...)
Affinity DataIC50:  27nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457385(CHEMBL4207561)
Affinity DataIC50:  27nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409053(6-(5-Fluoro-6-methylpyridin-3-yl)-3,3-dimethyl-1-(...)
Affinity DataIC50:  27nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457378(CHEMBL4203736)
Affinity DataIC50:  31nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409033(3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-1-(5-(meth...)
Affinity DataIC50:  32.1nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409050(1-(6-Cyclopropyl-5-(methylsulfonyl)pyridin-3-yl)-3...)
Affinity DataIC50:  38.5nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457384(CHEMBL4210157)
Affinity DataIC50:  39nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409044(1-(5-(Cyclopropylsulfonyl)pyridin-3-yl)-3,3-dimeth...)
Affinity DataIC50:  40nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409034(3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-1-(6-(meth...)
Affinity DataIC50:  40.1nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409037(5-(3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-2-oxoin...)
Affinity DataIC50:  44.9nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457376(CHEMBL4213616)
Affinity DataIC50:  52nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457377(CHEMBL4205790)
Affinity DataIC50:  57nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409049(5-(3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-2-oxoin...)
Affinity DataIC50:  71.7nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409048(5-(3,3-dimethyl-6-(2-methylpyrimidin-5-yl)-2-oxoin...)
Affinity DataIC50:  79.3nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457388(CHEMBL4217494)
Affinity DataIC50:  97nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409035(3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-1-(3-(meth...)
Affinity DataIC50:  106nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409046(5-(3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-2-oxoin...)
Affinity DataIC50:  128nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409043(1-(5-(Isopropylsulfonyl)pyridin-3-yl)-3,3-dimethyl...)
Affinity DataIC50:  135nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409055(3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-1-(5-(meth...)
Affinity DataIC50:  157nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409047(1-(5-(Azetidin-1-ylsulfonyl)pyridin-3-yl)-3,3-dime...)
Affinity DataIC50:  169nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409031(1-(Benzo[b]thiophen-6-yl)-3,3-dimethyl-6-(2-methyl...)
Affinity DataIC50:  189nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409051(3,3-Dimethyl-6-(2-methyl-1-oxidopyrimidin-1-ium-5-...)
Affinity DataIC50:  218nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409045(3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-1-(5-(meth...)
Affinity DataIC50:  218nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409056(6'-(2-Methylpyrimidin-5-yl)-1'-(5-(methylsulfonyl)...)
Affinity DataIC50:  230nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457380(CHEMBL4206265)
Affinity DataIC50:  244nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457383(CHEMBL4216732)
Affinity DataIC50:  253nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409052(3,3-Dimethyl-6-(5-methylpyridin-3-yl)-1-(5-(methyl...)
Affinity DataIC50:  313nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457382(CHEMBL4213885)
Affinity DataIC50:  321nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457389(CHEMBL4212469)
Affinity DataIC50:  838nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEquilibrative nucleoside transporter 1(Mus musculus (Mouse))
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409032(1-(Benzo[b]thiophen-4-yl)-3,3-dimethyl-6-(2-methyl...)
Affinity DataIC50:  844nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent