Compile Data Set for Download or QSAR
Found 15 of ic50 for UniProtKB: P31749
TargetRAC-alpha serine/threonine-protein kinase [E17K](Homo sapiens (Human))
TECHNISCHE UNIVERSITÄT DORTMUND

US Patent
LigandPNGBDBM50398379(CHEMBL2177390 | US10550114, Compound GDC-0068 | US...)
Affinity DataIC50:  2nMAssay Description:iFLiK and HTRF studies were carried out as described in Z. Fang, J. R. Simard, D. Plenker, H. D. Nguyen, T. Phan, P. Wolle, S. Baumeister, D. Rauh, A...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase [E17K](Homo sapiens (Human))
TECHNISCHE UNIVERSITÄT DORTMUND

US Patent
LigandPNGBDBM431867(US10550114, Compound 1a)
Affinity DataIC50:  80nMAssay Description:iFLiK and HTRF studies were carried out as described in Z. Fang, J. R. Simard, D. Plenker, H. D. Nguyen, T. Phan, P. Wolle, S. Baumeister, D. Rauh, A...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Homo sapiens (Human))
TECHNISCHE UNIVERSITÄT DORTMUND

US Patent
LigandPNGBDBM431879(US10550114, Compound 33)
Affinity DataIC50:  116nMAssay Description:iFLiK and HTRF studies were carried out as described in Z. Fang, J. R. Simard, D. Plenker, H. D. Nguyen, T. Phan, P. Wolle, S. Baumeister, D. Rauh, A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Homo sapiens (Human))
TECHNISCHE UNIVERSITÄT DORTMUND

US Patent
LigandPNGBDBM431885(US10550114, Compound 49)
Affinity DataIC50:  166nMAssay Description:iFLiK and HTRF studies were carried out as described in Z. Fang, J. R. Simard, D. Plenker, H. D. Nguyen, T. Phan, P. Wolle, S. Baumeister, D. Rauh, A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Homo sapiens (Human))
TECHNISCHE UNIVERSITÄT DORTMUND

US Patent
LigandPNGBDBM431884(US10550114, Compound 48)
Affinity DataIC50:  397nMAssay Description:iFLiK and HTRF studies were carried out as described in Z. Fang, J. R. Simard, D. Plenker, H. D. Nguyen, T. Phan, P. Wolle, S. Baumeister, D. Rauh, A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Homo sapiens (Human))
TECHNISCHE UNIVERSITÄT DORTMUND

US Patent
LigandPNGBDBM431877(US10550114, Compound 32)
Affinity DataIC50:  525nMAssay Description:iFLiK and HTRF studies were carried out as described in Z. Fang, J. R. Simard, D. Plenker, H. D. Nguyen, T. Phan, P. Wolle, S. Baumeister, D. Rauh, A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Homo sapiens (Human))
TECHNISCHE UNIVERSITÄT DORTMUND

US Patent
LigandPNGBDBM431882(US10550114, Compound 46)
Affinity DataIC50:  952nMAssay Description:iFLiK and HTRF studies were carried out as described in Z. Fang, J. R. Simard, D. Plenker, H. D. Nguyen, T. Phan, P. Wolle, S. Baumeister, D. Rauh, A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Homo sapiens (Human))
TECHNISCHE UNIVERSITÄT DORTMUND

US Patent
LigandPNGBDBM431881(US10550114, Compound 36)
Affinity DataIC50:  1.84E+3nMAssay Description:iFLiK and HTRF studies were carried out as described in Z. Fang, J. R. Simard, D. Plenker, H. D. Nguyen, T. Phan, P. Wolle, S. Baumeister, D. Rauh, A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Homo sapiens (Human))
TECHNISCHE UNIVERSITÄT DORTMUND

US Patent
LigandPNGBDBM431875(US10550114, Compound 30)
Affinity DataIC50:  1.95E+3nMAssay Description:iFLiK and HTRF studies were carried out as described in Z. Fang, J. R. Simard, D. Plenker, H. D. Nguyen, T. Phan, P. Wolle, S. Baumeister, D. Rauh, A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Homo sapiens (Human))
TECHNISCHE UNIVERSITÄT DORTMUND

US Patent
LigandPNGBDBM431886(US10550114, Compound 50)
Affinity DataIC50:  2.87E+3nMAssay Description:iFLiK and HTRF studies were carried out as described in Z. Fang, J. R. Simard, D. Plenker, H. D. Nguyen, T. Phan, P. Wolle, S. Baumeister, D. Rauh, A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Homo sapiens (Human))
TECHNISCHE UNIVERSITÄT DORTMUND

US Patent
LigandPNGBDBM431883(US10550114, Compound 47)
Affinity DataIC50:  2.90E+3nMAssay Description:iFLiK and HTRF studies were carried out as described in Z. Fang, J. R. Simard, D. Plenker, H. D. Nguyen, T. Phan, P. Wolle, S. Baumeister, D. Rauh, A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Homo sapiens (Human))
TECHNISCHE UNIVERSITÄT DORTMUND

US Patent
LigandPNGBDBM50313650(8-(4-(1-aminocyclobutyl)phenyl)-9-phenyl-[1,2,4]tr...)
Affinity DataIC50:  3.49E+3nMAssay Description:iFLiK and HTRF studies were carried out as described in Z. Fang, J. R. Simard, D. Plenker, H. D. Nguyen, T. Phan, P. Wolle, S. Baumeister, D. Rauh, A...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Homo sapiens (Human))
TECHNISCHE UNIVERSITÄT DORTMUND

US Patent
LigandPNGBDBM431876(US10550114, Compound 31)
Affinity DataIC50:  8.77E+3nMAssay Description:iFLiK and HTRF studies were carried out as described in Z. Fang, J. R. Simard, D. Plenker, H. D. Nguyen, T. Phan, P. Wolle, S. Baumeister, D. Rauh, A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Homo sapiens (Human))
TECHNISCHE UNIVERSITÄT DORTMUND

US Patent
LigandPNGBDBM431880(US10550114, Compound 45)
Affinity DataIC50:  2.37E+4nMAssay Description:iFLiK and HTRF studies were carried out as described in Z. Fang, J. R. Simard, D. Plenker, H. D. Nguyen, T. Phan, P. Wolle, S. Baumeister, D. Rauh, A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase [E17K](Homo sapiens (Human))
TECHNISCHE UNIVERSITÄT DORTMUND

US Patent
LigandPNGBDBM431874(US10550114, Compound 29)
Affinity DataIC50:  2.81E+4nMAssay Description:iFLiK and HTRF studies were carried out as described in Z. Fang, J. R. Simard, D. Plenker, H. D. Nguyen, T. Phan, P. Wolle, S. Baumeister, D. Rauh, A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent