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Found 10 of ki for UniProtKB: P15884
TargetTranscription factor 4(Homo sapiens)TBA
LigandPNGBDBM50509813(CHEMBL4451478)
Affinity DataKi:  640nMAssay Description:Inhibition of beta catenin/Tcf4 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranscription factor 4(Homo sapiens)TBA
LigandPNGBDBM50594243(CHEMBL5191974)
Affinity DataKi:  1.36E+3nMAssay Description:Binding affinity to beta-catenin (142 to 686 residues) (unknown origin)/C-terminal fluorescein-labeled human Tcf4 (7 to 51 residues) assessed as inhi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCatenin beta-1 [138-686]/Transcription factor 4 [7-51](Homo sapiens (Human))
University of Utah Research Foundation

US Patent
LigandPNGBDBM213761(US9284299, 12 | US9738628, Compound 12)
Affinity DataKi:  3.14E+3nM ΔG°:  -7.50kcal/moleT: 2°CAssay Description:Experiments were performed in 96-well Microfluor 2 black plates (Waltham, Mass.), and the samples were read by a Synergy 2 plate reader (Biotek, Wino...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCatenin beta-1 [138-686]/Transcription factor 4 [7-51](Homo sapiens (Human))
University of Utah Research Foundation

US Patent
LigandPNGBDBM32102(1,6-dimethylpyrimido[5,4-e][1,2,4]triazine-5,7(1H,...)
Affinity DataKi:  3.65E+3nM ΔG°:  -7.41kcal/molepH: 7.4 T: 2°CAssay Description:Experiments were performed in white opaque 384-well plates from PerkinElmer (Waltham, Mass.), and the samples were read on a Synergy 2 plate reader (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCatenin beta-1 [138-686]/Transcription factor 4 [7-51](Homo sapiens (Human))
University of Utah Research Foundation

US Patent
LigandPNGBDBM213761(US9284299, 12 | US9738628, Compound 12)
Affinity DataKi:  3.83E+3nM ΔG°:  -7.38kcal/molepH: 7.4 T: 2°CAssay Description:Experiments were performed in white opaque 384-well plates from PerkinElmer (Waltham, Mass.), and the samples were read on a Synergy 2 plate reader (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCatenin beta-1 [138-686]/Transcription factor 4 [7-51](Homo sapiens (Human))
University of Utah Research Foundation

US Patent
LigandPNGBDBM32102(1,6-dimethylpyrimido[5,4-e][1,2,4]triazine-5,7(1H,...)
Affinity DataKi:  5.82E+3nM ΔG°:  -7.14kcal/moleT: 2°CAssay Description:Experiments were performed in 96-well Microfluor 2 black plates (Waltham, Mass.), and the samples were read by a Synergy 2 plate reader (Biotek, Wino...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCatenin beta-1 [138-686]/Transcription factor 4 [7-51](Homo sapiens (Human))
University of Utah Research Foundation

US Patent
LigandPNGBDBM50094484(CHEBI:3556 | CHEMBL2323033 | US9284299, CGP049090 ...)
Affinity DataKi:  5.87E+3nM ΔG°:  -7.13kcal/molepH: 7.4 T: 2°CAssay Description:Experiments were performed in white opaque 384-well plates from PerkinElmer (Waltham, Mass.), and the samples were read on a Synergy 2 plate reader (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCatenin beta-1 [138-686]/Transcription factor 4 [7-51](Homo sapiens (Human))
University of Utah Research Foundation

US Patent
LigandPNGBDBM213748(US9284299, PKF115-584 | US9738628, Compound PKF115...)
Affinity DataKi:  1.78E+4nM ΔG°:  -6.48kcal/moleT: 2°CAssay Description:Experiments were performed in 96-well Microfluor 2 black plates (Waltham, Mass.), and the samples were read by a Synergy 2 plate reader (Biotek, Wino...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCatenin beta-1 [138-686]/Transcription factor 4 [7-51](Homo sapiens (Human))
University of Utah Research Foundation

US Patent
LigandPNGBDBM50094484(CHEBI:3556 | CHEMBL2323033 | US9284299, CGP049090 ...)
Affinity DataKi:  3.56E+4nM ΔG°:  -6.07kcal/moleT: 2°CAssay Description:Experiments were performed in 96-well Microfluor 2 black plates (Waltham, Mass.), and the samples were read by a Synergy 2 plate reader (Biotek, Wino...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTranscription factor 4(Homo sapiens)TBA
LigandPNGBDBM50094486(CHEMBL3589160)
Affinity DataKi:  7.60E+4nMAssay Description:Inhibition of beta catenin/Tcf4 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed