Compile Data Set for Download or QSAR
Report error Found 244 of ec50 for UniProtKB: P61073
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50225415BDBM50225415(WZ-811 | N,N'-di-2-pyridinyl-1,4-benzenedimethanam...)
Affinity DataEC50:  0.300nMAssay Description:Displacement of biotinylated TN14003 from CXCR4 in MDA-MB-231 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50102036BDBM50102036(Derivative of T140 peptide | CHEMBL2372985)
Affinity DataEC50:  0.400nMAssay Description:Effective concentration for 50% protection of HIV-induced cytopathogenicity in MT-4 cells on the MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50102035BDBM50102035(Derivative of T140 peptide | CHEMBL2372997)
Affinity DataEC50:  0.5nMAssay Description:Effective concentration for 50% protection of HIV-induced cytopathogenicity in MT-4 cells on the MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50102037BDBM50102037(Derivative of T140 peptide | CHEMBL2372993)
Affinity DataEC50:  0.600nMAssay Description:Effective concentration for 50% protection of HIV-induced cytopathogenicity in MT-4 cells on the MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50102047BDBM50102047(Derivative of T140 peptide | CHEMBL2373004)
Affinity DataEC50:  1.20nMAssay Description:Effective concentration for 50% protection of HIV-induced cytopathogenicity in MT-4 cells on the MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50102046BDBM50102046(Derivative of T140 peptide | CHEMBL2372989)
Affinity DataEC50:  2.70nMAssay Description:Effective concentration for 50% protection of HIV-induced cytopathogenicity in MT-4 cells on the MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403812BDBM50403812(CHEMBL2370108)
Affinity DataEC50:  2.80nMAssay Description:Inhibition of HIV-induced cytopathogenicity in MT-4 cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50102044BDBM50102044(Derivative of T140 peptide | CHEMBL2373002)
Affinity DataEC50:  2.80nMAssay Description:Effective concentration for 50% protection of HIV-induced cytopathogenicity in MT-4 cells on the MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096735BDBM50096735(Compound T140 | CHEMBL2372983)
Affinity DataEC50:  3.30nMAssay Description:Effective concentration for 50% protection of HIV-induced cytopathogenicity in MT-4 cells on the MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403817BDBM50403817(CHEMBL2370138)
Affinity DataEC50:  3.30nMAssay Description:Inhibition of HIV-induced cytopathogenicity in MT-4 cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403800BDBM50403800(TC-14004 | CHEMBL2370135)
Affinity DataEC50:  4nMAssay Description:Inhibition of HIV-induced cytopathogenicity in MT-4 cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50102040BDBM50102040(T140 | CHEMBL2372994)
Affinity DataEC50:  4nMAssay Description:Effective concentration for 50% protection of HIV-induced cytopathogenicity in MT-4 cells on the MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50327300BDBM50327300(CHEMBL1256528)
Affinity DataEC50:  4.40nMAssay Description:Displacement of [125I]-SDF-1-alpha from CXCR4 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50102032BDBM50102032(Derivative of T140 peptide | CHEMBL2373001)
Affinity DataEC50:  4.60nMAssay Description:Effective concentration for 50% protection of HIV-induced cytopathogenicity in MT-4 cells on the MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50102048BDBM50102048(Derivative of T140 peptide | CHEMBL2372999)
Affinity DataEC50:  6.60nMAssay Description:Effective concentration for 50% protection of HIV-induced cytopathogenicity in MT-4 cells on the MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50102034BDBM50102034(Derivative of T140 peptide | CHEMBL2372995)
Affinity DataEC50:  6.80nMAssay Description:Effective concentration for 50% protection of HIV-induced cytopathogenicity in MT-4 cells on the MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50327302BDBM50327302(CHEMBL1256583 | CHEMBL1256530)
Affinity DataEC50:  7.10nMAssay Description:Displacement of [125I]-SDF-1-alpha from CXCR4 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50327302BDBM50327302(CHEMBL1256583 | CHEMBL1256530)
Affinity DataEC50:  7.10nMAssay Description:Displacement of [125I]-SDF-1-alpha from CXCR4 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50102041BDBM50102041(Derivative of T140 peptide | CHEMBL2372990)
Affinity DataEC50:  7.80nMAssay Description:Effective concentration for 50% protection of HIV-induced cytopathogenicity in MT-4 cells on the MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50002692BDBM50002692(1-((2R,4S,5S)-4-Azido-5-hydroxymethyl-tetrahydro-f...)
Affinity DataEC50:  7.90nMAssay Description:Effective concentration for 50% protection of HIV-induced cytopathogenicity in MT-4 cells on the MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403809BDBM50403809(CHEMBL2370104)
Affinity DataEC50:  8.30nMAssay Description:Inhibition of HIV-induced cytopathogenicity in MT-4 cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50102038BDBM50102038(Derivative of T140 peptide | CHEMBL2372996)
Affinity DataEC50:  8.90nMAssay Description:Effective concentration for 50% protection of HIV-induced cytopathogenicity in MT-4 cells on the MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403810BDBM50403810(TC-14002 | CHEMBL2370137)
Affinity DataEC50:  9.30nMAssay Description:Inhibition of HIV-induced cytopathogenicity in MT-4 cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247595BDBM50247595(CHEMBL4064397)
Affinity DataEC50:  14nMAssay Description:Antagonist activity at CXCR4 in human CCRF-CEM cells assessed as inhibition of CXCL12-induced CXCR4+ cell migration pre-incubated for 10 mins before ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2019
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196276BDBM50196276(CHEMBL3982241)
Affinity DataEC50:  15nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403807BDBM50403807(CHEMBL2370130)
Affinity DataEC50:  15nMAssay Description:Inhibition of HIV-induced cytopathogenicity in MT-4 cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403806BDBM50403806(TC-14003 | CHEMBL2370132)
Affinity DataEC50:  15nMAssay Description:Inhibition of HIV-induced cytopathogenicity in MT-4 cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403815BDBM50403815(CHEMBL2370133)
Affinity DataEC50:  16nMAssay Description:Inhibition of HIV-induced cytopathogenicity in MT-4 cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403816BDBM50403816(CHEMBL2370136)
Affinity DataEC50:  16nMAssay Description:Inhibition of HIV-induced cytopathogenicity in MT-4 cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403805BDBM50403805(CHEMBL2370140)
Affinity DataEC50:  16nMAssay Description:Inhibition of HIV-induced cytopathogenicity in MT-4 cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403799BDBM50403799(CHEMBL2370105)
Affinity DataEC50:  17nMAssay Description:Inhibition of HIV-induced cytopathogenicity in MT-4 cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403801BDBM50403801(CHEMBL2370139)
Affinity DataEC50:  17nMAssay Description:Inhibition of HIV-induced cytopathogenicity in MT-4 cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403802BDBM50403802(TC-14007 | CHEMBL2370134)
Affinity DataEC50:  18nMAssay Description:Inhibition of HIV-induced cytopathogenicity in MT-4 cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50327301BDBM50327301(CHEMBL1256529)
Affinity DataEC50:  19nMAssay Description:Displacement of [125I]-SDF-1-alpha from CXCR4 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50102043BDBM50102043(Derivative of T140 peptide | CHEMBL2373005)
Affinity DataEC50:  36nMAssay Description:Effective concentration for 50% protection of HIV-induced cytopathogenicity in MT-4 cells on the MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50102042BDBM50102042(Derivative of T140 peptide | CHEMBL2373000)
Affinity DataEC50:  37nMAssay Description:Effective concentration for 50% protection of HIV-induced cytopathogenicity in MT-4 cells on the MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196260BDBM50196260(CHEMBL3914095)
Affinity DataEC50:  40nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50102045BDBM50102045(Derivative of T140 peptide | CHEMBL2373003)
Affinity DataEC50:  40nMAssay Description:Effective concentration for 50% protection of HIV-induced cytopathogenicity in MT-4 cells on the MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403818BDBM50403818(CHEMBL2370106)
Affinity DataEC50:  47nMAssay Description:Inhibition of HIV-induced cytopathogenicity in MT-4 cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50002692BDBM50002692(1-((2R,4S,5S)-4-Azido-5-hydroxymethyl-tetrahydro-f...)
Affinity DataEC50:  48nMAssay Description:Inhibition of HIV-induced cytopathogenicity in MT-4 cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196275BDBM50196275(CHEMBL3930215)
Affinity DataEC50:  50nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196257BDBM50196257(CHEMBL3903301)
Affinity DataEC50:  52nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403814BDBM50403814(CHEMBL3038227)
Affinity DataEC50:  56nMAssay Description:Inhibition of HIV-induced cytopathogenicity in MT-4 cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196240BDBM50196240(CHEMBL3896146)
Affinity DataEC50:  56nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196269BDBM50196269(CHEMBL3976727)
Affinity DataEC50:  58nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196270BDBM50196270(CHEMBL3963915)
Affinity DataEC50:  61nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196244BDBM50196244(CHEMBL3896065)
Affinity DataEC50:  62nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196251BDBM50196251(CHEMBL3912312)
Affinity DataEC50:  64nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50196262BDBM50196262(CHEMBL3978794)
Affinity DataEC50:  65nMAssay Description:Agonist activity at HA-tagged human CXCR4 receptor expressed in HEK293 cells co-transfected with Galphai1-91-RlucII, Gbeta1, and GFP10-G-gamma1 incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2018
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155310BDBM50155310(CHEMBL3779982)
Affinity DataEC50:  68nMAssay Description:Displacement of [125I]SDF-1 from human CXCR4 expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
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