Compile Data Set for Download or QSAR
maximum 50k data
Found 2 with your filter
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM138248(US8871738, 31)
Affinity DataIC50:  213nMAssay Description:Inhibition of recombinant CETP (unknown origin) assessed as inhibition of transfer of [3H]cholesteryl oleate or [3H]triolein between exogenous [3H]LD...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM138248(US8871738, 31)
Affinity DataIC50:  213nMpH: 7.4 T: 2°CAssay Description:First, low density lipoprotein (LDL) (Meridian) was biotinylated by incubating LDL with biotin for 1 hour on ice, after which it was dialyzed to remo...More data for this Ligand-Target Pair
In DepthDetails US Patent