Compile Data Set for Download or QSAR
maximum 50k data
Found 49 Enz. Inhib. hit(s) with all data for entry = 5780
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93394(PSTQ Analog, 3{1,27})
Affinity DataKi:  2.86nM IC50:  6.17nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93364(PSTQ Analog, 3{1,22})
Affinity DataKi:  3.54nM IC50:  7.62nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93393(PSTQ Analog, 3{1,26})
Affinity DataKi:  5.01nM IC50:  10.8nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93392(PSTQ Analog, 3{1,4})
Affinity DataKi:  7.04nM IC50:  15.2nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93385(PSTQ Analog, 3{1,43})
Affinity DataKi:  7.65nM IC50:  16.5nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93376(PSTQ Analog, 3{1,25})
Affinity DataKi:  12.9nM IC50:  27.8nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93363(PSTQ Analog, 3{1,21})
Affinity DataKi:  13.2nM IC50:  28.4nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93400(PSTQ Analog, 3{8,4})
Affinity DataKi:  16.7nM IC50:  35.9nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93399(PSTQ Analog, 3{1,49})
Affinity DataKi:  19.5nM IC50:  42.1nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93395(PSTQ Analog, 3{1,28})
Affinity DataKi:  27.6nM IC50:  59.5nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93391(PSTQ Analog, 3{1,3})
Affinity DataKi:  49.5nM IC50:  107nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93397(PSTQ Analog, 3{1,42})
Affinity DataIC50: >30nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93396(PSTQ Analog, 3{1,40})
Affinity DataIC50: >30nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93363(PSTQ Analog, 3{1,21})
Affinity DataIC50:  75.4nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93362(PSTQ Analog, 3{1,13})
Affinity DataIC50:  128nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93364(PSTQ Analog, 3{1,22})
Affinity DataIC50:  142nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93386(PSTQ Analog, 3{1,44})
Affinity DataIC50:  164nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93382(PSTQ Analog, 3{9,31})
Affinity DataIC50:  295nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93390(PSTQ Analog, 3{1,2})
Affinity DataIC50: >300nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93366(PSTQ Analog, 3{2,12})
Affinity DataIC50:  320nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93372(PSTQ Analog, 3{9,20})
Affinity DataIC50:  356nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93361(PSTQ Analog, 3{1,12})
Affinity DataIC50:  381nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93367(PSTQ Analog, 3{2,13})
Affinity DataIC50:  528nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93385(PSTQ Analog, 3{1,43})
Affinity DataIC50:  564nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93377(PSTQ Analog, 3{3,27})
Affinity DataIC50:  572nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93376(PSTQ Analog, 3{1,25})
Affinity DataIC50:  580nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93371(PSTQ Analog, 3{9,13})
Affinity DataIC50:  603nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93357(PSTQ Analog, 3{2,10})
Affinity DataIC50:  606nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93370(PSTQ Analog, 3{6,20})
Affinity DataIC50:  628nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93384(PSTQ Analog, 3{10,33})
Affinity DataIC50:  670nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93380(PSTQ Analog, 3{7,37})
Affinity DataIC50:  704nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93368(PSTQ Analog, 3{2,20})
Affinity DataIC50:  740nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93381(PSTQ Analog, 3{8,31})
Affinity DataIC50:  770nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93373(PSTQ Analog, 3{9,21})
Affinity DataIC50:  779nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93360(PSTQ Analog, 3{10,4})
Affinity DataIC50:  964nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93387(PSTQ Analog, 3{9,44})
Affinity DataIC50:  971nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93365(PSTQ Analog, 3{1,23})
Affinity DataIC50:  983nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93383(PSTQ Analog, 3{10,32})
Affinity DataIC50:  1.00E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93355(PSTQ Analog, 9)
Affinity DataIC50:  1.05E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93389(PSTQ Analog, 3{9,58})
Affinity DataIC50:  1.20E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93388(PSTQ Analog, 3{9,53})
Affinity DataIC50:  1.31E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93356(PSTQ Analog, 10)
Affinity DataIC50:  1.37E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93379(PSTQ Analog, 3{7,31})
Affinity DataIC50:  1.43E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93374(PSTQ Analog, 3{10,21})
Affinity DataIC50:  1.46E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93369(PSTQ Analog, 3{2,21})
Affinity DataIC50:  1.48E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93375(PSTQ Analog, 3{12,21})
Affinity DataIC50:  1.80E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93358(PSTQ Analog, 3{9,9})
Affinity DataIC50:  2.01E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93359(PSTQ Analog, 3{10,3})
Affinity DataIC50:  2.18E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Chemical Diversity Research Institute

LigandPNGBDBM93354(PSTQ Analog, 8)
Affinity DataIC50:  5.74E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed