Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 6073
TargetKiSS-1 receptor(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM107307(US8592379, 19)
Affinity DataIC50:  0.120nMAssay Description:Binding inhibition assay using human GPR54.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetKiSS-1 receptor(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM107314(US8592379, 36 | US8592379, 37)
Affinity DataIC50:  0.240nMAssay Description:Binding inhibition assay using human GPR54.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKiSS-1 receptor(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM107306(US8592379, 1)
Affinity DataIC50:  0.710nMAssay Description:Binding inhibition assay using human GPR54.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKiSS-1 receptor(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM107308(US8592379, 20)
Affinity DataIC50:  1.20nMAssay Description:Binding inhibition assay using human GPR54.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetKiSS-1 receptor(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM107309(US8592379, 21)
Affinity DataIC50:  4.60nMAssay Description:Binding inhibition assay using human GPR54.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetKiSS-1 receptor(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM107312(US8592379, 24a/24b | US8592379, 35)
Affinity DataIC50:  5.70nMAssay Description:Binding inhibition assay using human GPR54.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKiSS-1 receptor(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM107314(US8592379, 36 | US8592379, 37)
Affinity DataIC50:  32nMAssay Description:Binding inhibition assay using human GPR54.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKiSS-1 receptor(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM107310(US8592379, 22 | US8592379, 33)
Affinity DataIC50:  32nMAssay Description:Binding inhibition assay using human GPR54.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKiSS-1 receptor(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM107312(US8592379, 24a/24b | US8592379, 35)
Affinity DataIC50:  380nMAssay Description:Binding inhibition assay using human GPR54.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKiSS-1 receptor(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM47092(US8592379, 23)
Affinity DataIC50:  460nMAssay Description:Binding inhibition assay using human GPR54.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKiSS-1 receptor(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM107316(US8592379, 26)
Affinity DataIC50:  3.50E+3nMAssay Description:Binding inhibition assay using human GPR54.More data for this Ligand-Target Pair
In DepthDetails US Patent