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Found 17 Enz. Inhib. hit(s) with all data for entry = 6129
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM110223(US8618290, 61)
Affinity DataIC50:  3nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM110216(US8618290, 33)
Affinity DataIC50:  4nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM110229(US8618290, 85)
Affinity DataIC50:  4nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM110226(US8618290, 78)
Affinity DataIC50:  4nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM110221(US8618290, 58)
Affinity DataIC50:  5nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM110227(US8618290, 79)
Affinity DataIC50:  6nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM110218(US8618290, 37)
Affinity DataIC50:  6nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM110222(US8618290, 59)
Affinity DataIC50:  8nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM110228(US8618290, 83)
Affinity DataIC50:  8nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM110232(US8618290, 99)
Affinity DataIC50:  8nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM110230(US8618290, 93)
Affinity DataIC50:  8nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM110219(US8618290, 40)
Affinity DataIC50:  10nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM110224(US8618290, 65)
Affinity DataIC50:  10nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM110220(US8618290, 45)
Affinity DataIC50:  10nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM110225(US8618290, 75)
Affinity DataIC50:  10nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM110231(US8618290, 96)
Affinity DataIC50:  13nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM110217(US8618290, 35)
Affinity DataIC50:  13nMpH: 7.3Assay Description:An in vitro competition fluorescence polarization assay in which a test compound competes with a fluorescent probe for binding to the binding domain ...More data for this Ligand-Target Pair
In DepthDetails US Patent