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Found 11 Enz. Inhib. hit(s) with all data for entry = 50000340
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM591((2R,4S)-2-[(R)-(benzylcarbamoyl)(1-phenylacetamido...)
Affinity DataIC50:  0.900nMAssay Description:Inhibitory activity towards HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM589((2R,4S)-2-[(R)-carbamoyl(1-phenylacetamido)methyl]...)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity towards HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM590((2R,4S)-2-[(R)-(ethylcarbamoyl)(1-phenylacetamido)...)
Affinity DataIC50:  4.80nMAssay Description:Inhibitory activity towards HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM588(CHEMBL104525 | [ 2R-[ 2a(R*),4B ] ]-4,4 -[ 1,2-Eth...)
Affinity DataIC50:  60nMAssay Description:Inhibitory activity towards HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50004601((4-{2-[(3,3-Dimethyl-7-oxo-6-phenylacetylamino-4-t...)
Affinity DataIC50:  500nMAssay Description:Inhibitory activity towards HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50004600((4-{N'-[2-(Methoxycarbonyl-phenylacetylamino-methy...)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibitory activity towards HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50004598(CHEMBL322454 | [4-(3-{[2-(Methoxycarbonyl-phenylac...)
Affinity DataIC50: >1.20E+4nMAssay Description:Inhibitory activity towards HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50004602(2-[2-benzylcarboxamido(ethylcarbamoyl)methyl-5,5-d...)
Affinity DataIC50: >1.20E+4nMAssay Description:Inhibitory activity towards HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50004603(CHEMBL105589 | [4-(2-Acetylamino-ethylcarbamoyl)-5...)
Affinity DataIC50: >5.50E+4nMAssay Description:Inhibitory activity towards HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50004597((4-Ethylcarbamoyl-5,5-dimethyl-thiazolidin-2-yl)-p...)
Affinity DataIC50: >6.30E+4nMAssay Description:Inhibitory activity towards HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50004599(1N-[3-{2-[6-benzylcarboxamido-2,2-dimethyl-5-oxo-(...)
Affinity DataIC50: >7.00E+4nMAssay Description:Inhibitory activity towards HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed