Compile Data Set for Download or QSAR
maximum 50k data
Found 137 Enz. Inhib. hit(s) with all data for entry = 50001072
LigandPNGBDBM82376(CAS_80880-90-6 | NSC_5387 | TELENZEPINE)
Affinity DataKi:  1.80nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M1 of transfected rat A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012344(11-{2-[4-(10-Diethylamino-decyl)-piperazin-1-yl]-a...)
Affinity DataKi:  3nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M1 of transfected A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012336(11-(2-{4-[10-(2-Methoxy-benzylamino)-decyl]-pipera...)
Affinity DataKi:  3.30nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M1 of transfected A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM82376(CAS_80880-90-6 | NSC_5387 | TELENZEPINE)
Affinity DataKi:  6.90nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M3 of transfected rat A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012353(11-{2-[4-(10-Amino-decyl)-piperazin-1-yl]-acetyl}-...)
Affinity DataKi:  12nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M2 of rat heart tissue membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012344(11-{2-[4-(10-Diethylamino-decyl)-piperazin-1-yl]-a...)
Affinity DataKi:  14nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M2 of rat heart tissue membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012353(11-{2-[4-(10-Amino-decyl)-piperazin-1-yl]-acetyl}-...)
Affinity DataKi:  16nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M1 of transfected A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM82376(CAS_80880-90-6 | NSC_5387 | TELENZEPINE)
Affinity DataKi:  17nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to muscarinic acetylcholine receptor M4 of rat heart NG108-15 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012348(2-(6-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido...)
Affinity DataKi:  18nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M2 of rat heart tissue membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012348(2-(6-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido...)
Affinity DataKi:  18nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M1 of transfected A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012360(11-{2-[4-(8-Amino-octyl)-piperazin-1-yl]-acetyl}-5...)
Affinity DataKi:  20nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M1 of transfected A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012357(2-(5-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido...)
Affinity DataKi:  20nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M2 of rat heart tissue membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012338((6-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido[3...)
Affinity DataKi:  21nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M2 of rat heart tissue membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012336(11-(2-{4-[10-(2-Methoxy-benzylamino)-decyl]-pipera...)
Affinity DataKi:  22nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M2 of rat heart tissue membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012338((6-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido[3...)
Affinity DataKi:  23nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to muscarinic acetylcholine receptor M4 of rat heart NG108-15 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012345(11-{2-[4-(9-Amino-nonyl)-piperazin-1-yl]-acetyl}-5...)
Affinity DataKi:  24nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M2 of rat heart tissue membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012345(11-{2-[4-(9-Amino-nonyl)-piperazin-1-yl]-acetyl}-5...)
Affinity DataKi:  24nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M1 of transfected A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012360(11-{2-[4-(8-Amino-octyl)-piperazin-1-yl]-acetyl}-5...)
Affinity DataKi:  26nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M2 of rat heart tissue membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  29nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M1 of transfected rat A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012338((6-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido[3...)
Affinity DataKi:  37nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M1 of transfected rat A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012371(CHEMBL70154 | N-(10-{4-[2-Oxo-2-(6-oxo-5,6-dihydro...)
Affinity DataKi:  43nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M2 of rat heart tissue membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012338((6-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido[3...)
Affinity DataKi:  46nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M3 of transfected rat A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM82376(CAS_80880-90-6 | NSC_5387 | TELENZEPINE)
Affinity DataKi:  50nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M2 of rat heart tissue membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012327(CHEMBL68292 | N-(9-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-...)
Affinity DataKi:  50nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M2 of rat heart tissue membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012365(11-{2-[4-(2-Chloro-ethyl)-piperazin-1-yl]-acetyl}-...)
Affinity DataKi:  52nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M1 of transfected A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012327(CHEMBL68292 | N-(9-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-...)
Affinity DataKi:  52nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M1 of transfected A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012351(11-{2-[4-(7-Amino-heptyl)-piperazin-1-yl]-acetyl}-...)
Affinity DataKi:  57nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M2 of rat heart tissue membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012357(2-(5-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido...)
Affinity DataKi:  60nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M1 of transfected rat A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012351(11-{2-[4-(7-Amino-heptyl)-piperazin-1-yl]-acetyl}-...)
Affinity DataKi:  66nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M1 of transfected A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012371(CHEMBL70154 | N-(10-{4-[2-Oxo-2-(6-oxo-5,6-dihydro...)
Affinity DataKi:  75nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M1 of transfected A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012365(11-{2-[4-(2-Chloro-ethyl)-piperazin-1-yl]-acetyl}-...)
Affinity DataKi:  78nMAssay Description:The compound was tested for the inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M3 of transfected A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012331(2-(4-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido...)
Affinity DataKi:  89nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M2 of rat heart tissue membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012331(2-(4-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido...)
Affinity DataKi:  120nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M3 of transfected rat A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012365(11-{2-[4-(2-Chloro-ethyl)-piperazin-1-yl]-acetyl}-...)
Affinity DataKi:  130nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M4 of NG108-15 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012331(2-(4-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido...)
Affinity DataKi:  170nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M1 of transfected rat A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012331(2-(4-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido...)
Affinity DataKi:  210nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to muscarinic acetylcholine receptor M4 of rat heart NG108-15 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012365(11-{2-[4-(2-Chloro-ethyl)-piperazin-1-yl]-acetyl}-...)
Affinity DataKi:  210nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M2 of rat heart tissue membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012340(11-[2-(4-Benzyl-piperazin-1-yl)-acetyl]-5,11-dihyd...)
Affinity DataKi:  220nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to muscarinic acetylcholine receptor M4 of rat heart NG108-15 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012340(11-[2-(4-Benzyl-piperazin-1-yl)-acetyl]-5,11-dihyd...)
Affinity DataKi:  240nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M3 of transfected rat A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012340(11-[2-(4-Benzyl-piperazin-1-yl)-acetyl]-5,11-dihyd...)
Affinity DataKi:  240nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M2 of rat heart tissue membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  240nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M3 of transfected rat A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012340(11-[2-(4-Benzyl-piperazin-1-yl)-acetyl]-5,11-dihyd...)
Affinity DataKi:  330nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M1 of transfected rat A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  330nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to muscarinic acetylcholine receptor M4 of rat heart NG108-15 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50406547(CHEMBL2112217)
Affinity DataKi:  370nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M1 of transfected rat A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  610nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M2 of rat heart tissue membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012346(CHEMBL70003 | N-(2-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-...)
Affinity DataKi:  670nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M1 of transfected rat A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012349(2-(3-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido...)
Affinity DataKi:  840nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M2 of rat heart tissue membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012363(CHEMBL305403 | N-(2-Amino-ethyl)-4-{4-[2-oxo-2-(6-...)
Affinity DataKi:  960nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M2 of rat heart tissue membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012346(CHEMBL70003 | N-(2-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-...)
Affinity DataKi:  970nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M3 of transfected rat A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012363(CHEMBL305403 | N-(2-Amino-ethyl)-4-{4-[2-oxo-2-(6-...)
Affinity DataKi:  1.04E+3nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to muscarinic acetylcholine receptor M4 of rat heart NG108-15 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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