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Found 12 Enz. Inhib. hit(s) with all data for entry = 50002268
TargetGamma-aminobutyric acid receptor subunit gamma-1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50021185(5-Aminomethyl-4,5-dihydro-isoxazol-3-ol | CHEMBL42...)
Affinity DataIC50:  4nMAssay Description:In vitro inhibition of [3H]-GABA binding to Gamma-aminobutyric-acid receptor of rat brain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit gamma-1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM23183(5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL2...)
Affinity DataIC50:  6nMAssay Description:In vitro inhibition of [3H]-GABA binding to Gamma-aminobutyric-acid receptor of rat brain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit gamma-1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...)
Affinity DataIC50:  33nMAssay Description:In vitro inhibition of [3H]-GABA binding to Gamma-aminobutyric-acid receptor of rat brain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit gamma-1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50021189(5-Aminomethyl-4,5-dihydro-isoxazol-3-ol | CHEMBL40...)
Affinity DataIC50:  250nMAssay Description:In vitro inhibition of [3H]-GABA binding to Gamma-aminobutyric-acid receptor of rat brain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit gamma-1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50021186(4-Amino-3-hydroxy-butyric acid | CHEMBL296263 | S(...)
Affinity DataIC50:  400nMAssay Description:In vitro inhibition of [3H]-GABA binding to Gamma-aminobutyric-acid receptor of rat brain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...)
Affinity DataIC50:  3.00E+3nMAssay Description:In vitro inhibition of GABA uptake in rat brain synaptic membranesMore data for this Ligand-Target Pair
LigandPNGBDBM50021186(4-Amino-3-hydroxy-butyric acid | CHEMBL296263 | S(...)
Affinity DataIC50:  2.90E+4nMAssay Description:In vitro inhibition of GABA uptake in rat brain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50021187(4-Amino-3-hydroxy-butyric acid | CHEMBL290216 | R(...)
Affinity DataIC50:  6.70E+4nMAssay Description:In vivo inhibition of GABA uptake in rat brain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50021189(5-Aminomethyl-4,5-dihydro-isoxazol-3-ol | CHEMBL40...)
Affinity DataIC50:  7.00E+4nMAssay Description:In vivo inhibition of GABA uptake in rat brain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225363(CHEMBL40363)
Affinity DataIC50:  1.30E+5nMAssay Description:In vitro inhibition of GABA uptake in rat brain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM23183(5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL2...)
Affinity DataIC50:  3.20E+5nMAssay Description:In vitro inhibition of GABA uptake in rat brain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50021185(5-Aminomethyl-4,5-dihydro-isoxazol-3-ol | CHEMBL42...)
Affinity DataIC50: >5.00E+5nMAssay Description:In vitro inhibition of GABA uptake in rat brain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed