Compile Data Set for Download or QSAR
maximum 50k data
Found 47 Enz. Inhib. hit(s) with all data for entry = 50036002
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002533(2-[2-(2-tert-Butoxycarbonylamino-4-carbamoyl-butyr...)
Affinity DataIC50:  90nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002552(CHEMBL303337 | benzyl 2-[2-(1-formyl-1H-3-indolyl)...)
Affinity DataIC50:  110nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002568(CHEMBL304472 | benzyl 2-[2-(1-formyl-1H-3-indolyl)...)
Affinity DataIC50:  110nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002543(CHEMBL59615 | benzyl 2-[2-[3-carbamoyl-1-neopentyl...)
Affinity DataIC50:  140nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002562(CHEMBL294798 | benzyl 2-[1-[3-carbamoyl-1-neopenty...)
Affinity DataIC50:  140nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002545(CHEMBL544284 | benzyl 2-[1-[1-amino-3-carbamoyl-(1...)
Affinity DataIC50:  210nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002571(CHEMBL293355 | benzyl 2-[1-[3-carbamoyl-1-neopenty...)
Affinity DataIC50:  240nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002573(CHEMBL58245 | benzyl 2-[2-(1-formyl-1H-3-indolyl)-...)
Affinity DataIC50:  260nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002563(CHEMBL62357 | benzyl 2-[1-[3-carbamoyl-1-neopentyl...)
Affinity DataIC50:  360nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002560(CHEMBL294814 | benzyl 2-[1-[3-carbamoyl-1-neopenty...)
Affinity DataIC50:  380nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002575(CHEMBL64166 | benzyl 2-[1-[3-carbamoyl-1-neopentyl...)
Affinity DataIC50:  390nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002564(Benzyloxycarbonyl-Gln-D-Trp(CHO)-Phe(methoxy-cyclo...)
Affinity DataIC50:  400nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002555(CHEMBL293726 | benzyl 2-[2-(1-formyl-1H-3-indolyl)...)
Affinity DataIC50:  420nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002570(CHEMBL417390 | benzyl 2-benzoyl-1-[2-[3-carbamoyl-...)
Affinity DataIC50:  450nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002557(Benzyloxycarbonyl-Gln-D-Trp(CHO)-Phe(ethoxyphenyl)...)
Affinity DataIC50:  500nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002536(CHEMBL292320 | benzyl 2-[1-[3-carbamoyl-1-neopenty...)
Affinity DataIC50:  550nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002539(CHEMBL405795 | D-Pro-Gln-Gln-D-Trp-Phe-D-Trp-D-Trp...)
Affinity DataIC50:  600nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002548(CHEMBL304246 | benzyl 2-[1-[3-carbamoyl-1-neopenty...)
Affinity DataIC50:  770nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002576(CHEMBL303543 | benzyl 2-[1-[3-carbamoyl-1-neopenty...)
Affinity DataIC50:  790nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002551(CHEMBL59768 | benzyl 2-[1-[3-carbamoyl-1-neopentyl...)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002556(Benzyloxycarbonyl-Gln-D-Trp(CHO)-Phe(4-chloro-meth...)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002532(CHEMBL63059 | benzyl 2-[1-[3-carbamoyl-1-neopentyl...)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002530(Benzyloxycarbonyl-Gln-D-Trp(CHO)-Phe(isopropyloxy)...)
Affinity DataIC50:  1.70E+3nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002550(Benzyloxycarbonyl-Phe-D-Trp-D-Trp-amine | CHEMBL62...)
Affinity DataIC50:  2.50E+3nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002540(Benzyloxycarbonyl-Gln-D-Trp(CHO)-Phe(methoxy) | CH...)
Affinity DataIC50:  1.00E+4nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002544(CHEMBL294288 | benzyl 2-[1-[3-carbamoyl-1-neopenty...)
Affinity DataIC50:  1.00E+4nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002531(CHEMBL62349 | benzyl 3-(1H-3-indolyl)-2-[1-[2-(1H-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002547(1N-[1-[1-carbamoyl-2-phenyl-(1S)-ethylcarbamoyl]-2...)
Affinity DataIC50:  1.00E+4nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002561(CHEMBL64631 | benzyl 2-[1-[1-benzyloxycarbonyl-(5R...)
Affinity DataIC50:  1.00E+4nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002549(CHEMBL64037 | tert-butyloxycarbonyl-D-Trp-D-Trp-Ph...)
Affinity DataIC50:  1.76E+4nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002558(Benzyloxycarbonyl-D-Trp-Phe-D-Trp-OH | CHEMBL30266...)
Affinity DataIC50:  2.38E+4nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002574(CHEMBL263013 | tert-butyloxycarbonyl-Gln-D-Trp-Phe...)
Affinity DataIC50:  3.87E+4nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002572(2-[1-[1-amino-2-phenyl-(1S)-ethylcarboxamido]-2-(1...)
Affinity DataIC50:  5.80E+4nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002542(CHEMBL64806 | tert-butyloxycarbonyl-Gln-D-Trp-Phe-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002534(Benzyloxycarbonyl-D-Trp-Phe-D-Trp-amine | CHEMBL30...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002537(Benzyloxycarbonyl-D-Pro-Gln-Gln-amine | CHEMBL2916...)
Affinity DataIC50:  1.00E+5nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002554(2-[3-carbamoyl-1-[2-oxo-(5S)-dihydro-1H-5-pyrrolyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002553(Benzyloxycarbonyl-D-Pro-Gln-Gln-OH | CHEMBL293179)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002567(2-[1-[1-amino-2-(1H-3-indolyl)-(1R)-ethylcarboxami...)
Affinity DataIC50:  1.00E+5nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002569(Benzyloxycarbonyl-Phe-D-Trp-D-Trp-OH | CHEMBL62634)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002546(4-carbamoyl-2-[3-carbamoyl-1-[(5R)-dihydro-1H-5-py...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002565(CHEMBL293200 | benzyl 2-[2-(1H-3-indolyl)-1-[2-(1H...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002566(CHEMBL293445 | benzyl 3-(1H-3-indolyl)-2-[2-(1H-3-...)
Affinity DataIC50:  1.00E+5nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002541(CHEMBL64829 | tert-butyl 5-[1-[1-benzyloxycarbonyl...)
Affinity DataIC50:  1.00E+5nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002538(CHEMBL294065 | tert-butyloxycarbonyl-Gln-D-Trp(CHO...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002535(2-[2-(1-methyl-1H-3-indolyl)-1-[2-oxo-(5S)-dihydro...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002559(CHEMBL304702 | tert-butyl 5-[3-carbamoyl-1-[1,3-di...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed