Compile Data Set for Download or QSAR
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Found 18 Enz. Inhib. hit(s) with all data for entry = 50036229
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50041573(17-(cyclopropylmethyl)-17'-butyl-6,6',7,7'-tetrade...)
Affinity DataKi:  0.0400nMAssay Description:The binding affinity on kappa-opioid receptor using [3H]- U-69,593 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM82551(C18130 | CAS_105618-26-6 | NOR-BNI (HCI)2 | NORBNI)
Affinity DataKi:  0.280nMAssay Description:The binding affinity on kappa-opioid receptor using [3H]- U-69,593 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50041568(17-(cyclopropylmethyl)-17'-[2-[(carbobenzyloxy)ami...)
Affinity DataKi:  0.360nMAssay Description:The binding affinity on kappa-opioid receptor using [3H]- U-69,593 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50041572(17-(cyclopropylmethyl)-17'-(2-guanidinoethyl-6,6',...)
Affinity DataKi:  0.590nMAssay Description:The binding affinity on kappa-opioid receptor using [3H]- U-69,593 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50041570(17-(cyclopropylmethyl)-17'-aminoethyl-6,6',7,7'-te...)
Affinity DataKi:  3.40nMAssay Description:The binding affinity on kappa-opioid receptor using [3H]- U-69,593 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50041573(17-(cyclopropylmethyl)-17'-butyl-6,6',7,7'-tetrade...)
Affinity DataKi:  15nMAssay Description:The binding affinity on delta-opioid receptor using [3H]- DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50041569(17-(cyclopropylmethyl)-17'-aminoethyl-6,6',7,7'-te...)
Affinity DataKi:  21nMAssay Description:The binding affinity on kappa-opioid receptor using [3H]- U-69,593 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50041572(17-(cyclopropylmethyl)-17'-(2-guanidinoethyl-6,6',...)
Affinity DataKi:  37nMAssay Description:The binding affinity on delta-opioid receptor using [3H]- DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM82551(C18130 | CAS_105618-26-6 | NOR-BNI (HCI)2 | NORBNI)
Affinity DataKi:  43nMAssay Description:The binding affinity on delta-opioid receptor using [3H]- DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50041570(17-(cyclopropylmethyl)-17'-aminoethyl-6,6',7,7'-te...)
Affinity DataKi:  46nMAssay Description:The binding affinity against mu-opioid receptor using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM82551(C18130 | CAS_105618-26-6 | NOR-BNI (HCI)2 | NORBNI)
Affinity DataKi:  47nMAssay Description:The binding affinity against mu-opioid receptor using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50041572(17-(cyclopropylmethyl)-17'-(2-guanidinoethyl-6,6',...)
Affinity DataKi:  50nMAssay Description:The binding affinity against mu-opioid receptor using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50041569(17-(cyclopropylmethyl)-17'-aminoethyl-6,6',7,7'-te...)
Affinity DataKi:  66nMAssay Description:The binding affinity against mu-opioid receptor using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50041568(17-(cyclopropylmethyl)-17'-[2-[(carbobenzyloxy)ami...)
Affinity DataKi:  70nMAssay Description:The binding affinity against mu-opioid receptor using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50041573(17-(cyclopropylmethyl)-17'-butyl-6,6',7,7'-tetrade...)
Affinity DataKi:  73nMAssay Description:The binding affinity against mu-opioid receptor using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50041568(17-(cyclopropylmethyl)-17'-[2-[(carbobenzyloxy)ami...)
Affinity DataKi:  117nMAssay Description:The binding affinity on delta-opioid receptor using [3H]- DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50041570(17-(cyclopropylmethyl)-17'-aminoethyl-6,6',7,7'-te...)
Affinity DataKi:  137nMAssay Description:The binding affinity on delta-opioid receptor using [3H]- DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50041569(17-(cyclopropylmethyl)-17'-aminoethyl-6,6',7,7'-te...)
Affinity DataKi: >1.00E+3nMAssay Description:The binding affinity on delta-opioid receptor using [3H]- DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed