Affinity DataIC50: 800nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40E+3nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+4nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+4nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+4nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+4nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 4.50E+4nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40E+4nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 5.80E+4nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+4nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 7.20E+4nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+4nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 9.50E+4nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+5nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+5nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+5nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+5nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+5nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+5nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+5nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+5nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+5nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+5nMAssay Description:Antagonism of adenosine A1 receptor assessed from the ability to inhibit binding of [3H]-cyclohexyladenosine to rat cerebral cortical membranesMore data for this Ligand-Target Pair