TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 0.0200nMAssay Description:Tested for inhibitory effect on binding of [3H]bremazocine to opioid receptor kappa in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 0.0290nMAssay Description:Tested for inhibitory effect on binding of [3H]bremazocine to opioid receptor kappa in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 0.0300nMAssay Description:Tested for inhibitory effect on binding of [3H]bremazocine to opioid receptor kappa in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 0.0490nMAssay Description:Tested for inhibitory effect on binding of [3H]bremazocine to opioid receptor kappa in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Tested for inhibitory effect on binding of [3H]DAMGO to opioid receptor mu in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Tested for inhibitory effect on binding of [3H]bremazocine to opioid receptor kappa in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Tested for inhibitory effect on binding of [3H]bremazocine to opioid receptor kappa in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Tested for inhibitory effect on binding of [3H]DPDPE to opioid receptor delta in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataKi: 3.60nMAssay Description:Tested for inhibitory effect on binding of [3H]bremazocine to opioid receptor kappa in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 9.60nMAssay Description:Tested for inhibitory effect on binding of [3H]DAMGO to opioid receptor mu in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Tested for inhibitory effect on binding of [3H]DAMGO to opioid receptor mu in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Tested for inhibitory effect on binding of [3H]DAMGO to opioid receptor mu in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Tested for inhibitory effect on binding of [3H]DAMGO to opioid receptor mu in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 149nMAssay Description:Tested for inhibitory effect on binding of [3H]DPDPE to opioid receptor delta in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 176nMAssay Description:Tested for inhibitory effect on binding of [3H]DPDPE to opioid receptor delta in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 206nMAssay Description:Tested for inhibitory effect on binding of [3H]DAMGO to opioid receptor mu in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 449nMAssay Description:Tested for inhibitory effect on binding of [3H]DPDPE to opioid receptor delta in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 551nMAssay Description:Tested for inhibitory effect on binding of [3H]DAMGO to opioid receptor mu in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 558nMAssay Description:Tested for inhibitory effect on binding of [3H]DPDPE to opioid receptor delta in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Homo sapiens (Human))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataIC50: 0.220nMAssay Description:Tested for opioid receptor agonistic activity in guinea pig ileumMore data for this Ligand-Target Pair
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Homo sapiens (Human))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Tested for opioid receptor agonistic activity in guinea pig ileumMore data for this Ligand-Target Pair
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Homo sapiens (Human))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataIC50: 2.60nMAssay Description:Tested for opioid receptor agonistic activity in guinea pig ileumMore data for this Ligand-Target Pair
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Homo sapiens (Human))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Tested for inhibitory effect on binding of [3H]DAMGO to opioid receptor mu in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Homo sapiens (Human))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataIC50: 687nMAssay Description:Tested for inhibitory effect on binding of [3H]bremazocine to opioid receptor kappa in guinea pig cerebellum membranesMore data for this Ligand-Target Pair
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Homo sapiens (Human))
Oregon State University
Curated by ChEMBL
Oregon State University
Curated by ChEMBL
Affinity DataIC50: 990nMAssay Description:Tested for opioid receptor agonistic activity in guinea pig ileumMore data for this Ligand-Target Pair