Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Inhibition of (unknown origin) 17beta-HSD1 assessed as conversion of [14C]estradiol to [14C]estrone using NADP+More data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of 17beta-HSD1 expressed in HEK 293 cells assessed as conversion of [14C]estrone to [14C]estradiol using NADPHMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of (unknown origin) 17beta-HSD1 expressed in HEK 293 cells assessed as conversion of [14C]estrone to [14C]estradiol using NADHMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Affinity DataIC50: 93nMAssay Description:Inhibition of (unknown origin) 17beta-HSD1 expressed in HEK 293 cells assessed as conversion of [14C]estrone to [14C]estradiol using NADHMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of (unknown origin) 17beta-HSD1 expressed in HEK 293 cells assessed as conversion of [14C]estrone to [14C]estradiolMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of (unknown origin) 17beta-HSD1 expressed in HEK 293 cells assessed as conversion of [14C]estrone to [14C]estradiolMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Affinity DataIC50: 310nMAssay Description:Inhibition of (unknown origin) 17beta-HSD1 expressed in HEK 293 cells assessed as conversion of [14C]estrone to [14C]estradiolMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Inhibition of (unknown origin) 17beta-HSD1 expressed in HEK 293 cells assessed as conversion of [14C]estrone to [14C]estradiol using NADHMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of (unknown origin) 17beta-HSD1 expressed in HEK 293 cells assessed as conversion of [14C]estrone to [14C]estradiolMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Affinity DataIC50: 810nMAssay Description:Inhibition of (unknown origin) 17beta-HSD1 expressed in HEK 293 cells assessed as conversion of [14C]estrone to [14C]estradiol using NADHMore data for this Ligand-Target Pair
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Chuq-Pavillon Chul And Université
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of (unknown origin) 17beta-HSD1 expressed in HEK 293 cells assessed as conversion of [14C]estrone to [14C]estradiol using NADHMore data for this Ligand-Target Pair