Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50044909
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Pharmacology And Toxicology

Curated by ChEMBL
LigandPNGBDBM50035854(CHEMBL3360487)
Affinity DataIC50:  8.70E+5nMAssay Description:Inhibition of human acetylcholinesterase by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Pharmacology And Toxicology

Curated by ChEMBL
LigandPNGBDBM50399977(CHEMBL2181432)
Affinity DataIC50:  8.90E+5nMAssay Description:Inhibition of human acetylcholinesterase by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Pharmacology And Toxicology

Curated by ChEMBL
LigandPNGBDBM50035853(CHEMBL3360486)
Affinity DataIC50:  9.30E+5nMAssay Description:Inhibition of human acetylcholinesterase by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Pharmacology And Toxicology

Curated by ChEMBL
LigandPNGBDBM50035852(HI-6)
Affinity DataIC50:  1.36E+6nMAssay Description:Inhibition of human acetylcholinesterase by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Pharmacology And Toxicology

Curated by ChEMBL
LigandPNGBDBM50333779(1,3-Bis(4-(Hydroxyimino-methyl)-pyridinium)-2-oxap...)
Affinity DataIC50:  2.21E+6nMAssay Description:Inhibition of human acetylcholinesterase by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Pharmacology And Toxicology

Curated by ChEMBL
LigandPNGBDBM50041520(1,3-PROPYLENE-BIS-N,N''-SYN-4-PYRIDINIUMALDOXIME |...)
Affinity DataIC50:  2.57E+6nMAssay Description:Inhibition of human acetylcholinesterase by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Pharmacology And Toxicology

Curated by ChEMBL
LigandPNGBDBM50399977(CHEMBL2181432)
Affinity DataKd:  2.20E+4nMAssay Description:Reactivation of VX-inhibited human acetylcholinesterase assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Pharmacology And Toxicology

Curated by ChEMBL
LigandPNGBDBM50035853(CHEMBL3360486)
Affinity DataKd:  2.40E+4nMAssay Description:Reactivation of VX-inhibited human acetylcholinesterase assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Pharmacology And Toxicology

Curated by ChEMBL
LigandPNGBDBM50035854(CHEMBL3360487)
Affinity DataKd:  2.50E+4nMAssay Description:Reactivation of VX-inhibited human acetylcholinesterase assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Pharmacology And Toxicology

Curated by ChEMBL
LigandPNGBDBM50333779(1,3-Bis(4-(Hydroxyimino-methyl)-pyridinium)-2-oxap...)
Affinity DataKd:  6.60E+4nMAssay Description:Reactivation of tabun-inhibited human acetylcholinesterase assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Pharmacology And Toxicology

Curated by ChEMBL
LigandPNGBDBM50041520(1,3-PROPYLENE-BIS-N,N''-SYN-4-PYRIDINIUMALDOXIME |...)
Affinity DataKd:  7.90E+4nMAssay Description:Reactivation of tabun-inhibited human acetylcholinesterase assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Pharmacology And Toxicology

Curated by ChEMBL
LigandPNGBDBM50399977(CHEMBL2181432)
Affinity DataKd:  1.80E+4nMAssay Description:Reactivation of tabun-inhibited human acetylcholinesterase assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Pharmacology And Toxicology

Curated by ChEMBL
LigandPNGBDBM50035853(CHEMBL3360486)
Affinity DataKd:  2.60E+4nMAssay Description:Reactivation of tabun-inhibited human acetylcholinesterase assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Pharmacology And Toxicology

Curated by ChEMBL
LigandPNGBDBM50035854(CHEMBL3360487)
Affinity DataKd:  1.40E+4nMAssay Description:Reactivation of tabun-inhibited human acetylcholinesterase assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Pharmacology And Toxicology

Curated by ChEMBL
LigandPNGBDBM50035852(HI-6)
Affinity DataKd:  2.70E+4nMAssay Description:Reactivation of VX-inhibited human acetylcholinesterase assessed as dissociation constantMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Pharmacology And Toxicology

Curated by ChEMBL
LigandPNGBDBM50333779(1,3-Bis(4-(Hydroxyimino-methyl)-pyridinium)-2-oxap...)
Affinity DataKd:  3.20E+4nMAssay Description:Reactivation of VX-inhibited human acetylcholinesterase assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Pharmacology And Toxicology

Curated by ChEMBL
LigandPNGBDBM50035854(CHEMBL3360487)
Affinity DataKd:  4.10E+4nMAssay Description:Reactivation of sarin-inhibited human acetylcholinesterase assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Pharmacology And Toxicology

Curated by ChEMBL
LigandPNGBDBM50035853(CHEMBL3360486)
Affinity DataKd:  1.43E+5nMAssay Description:Reactivation of sarin-inhibited human acetylcholinesterase assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Pharmacology And Toxicology

Curated by ChEMBL
LigandPNGBDBM50399977(CHEMBL2181432)
Affinity DataKd:  8.80E+4nMAssay Description:Reactivation of sarin-inhibited human acetylcholinesterase assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Pharmacology And Toxicology

Curated by ChEMBL
LigandPNGBDBM50333779(1,3-Bis(4-(Hydroxyimino-methyl)-pyridinium)-2-oxap...)
Affinity DataKd:  9.00E+4nMAssay Description:Reactivation of sarin-inhibited human acetylcholinesterase assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Pharmacology And Toxicology

Curated by ChEMBL
LigandPNGBDBM50035852(HI-6)
Affinity DataKd:  9.30E+4nMAssay Description:Reactivation of sarin-inhibited human acetylcholinesterase assessed as dissociation constantMore data for this Ligand-Target Pair