Affinity DataKi: 0.110nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.210nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.390nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.390nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.780nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibitory activity against CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibitory activity against CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 510nMAssay Description:Inhibitory activity against CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 530nMAssay Description:Inhibitory activity against CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 670nMAssay Description:Inhibitory activity against CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 760nMAssay Description:Inhibitory activity against CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibitory activity against CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibitory activity against CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory activity against CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibitory activity against CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibitory activity against CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory activity against CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 8.70E+3nMAssay Description:Inhibitory activity against CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibitory activity against CYP2D6More data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Agonist activity at kappa opioid receptor in a [35S]GTPgammaS functional assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.230nMAssay Description:Agonist activity at kappa opioid receptor in a [35S]GTPgammaS functional assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.230nMAssay Description:Agonist activity at kappa opioid receptor in a [35S]GTPgammaS functional assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.800nMAssay Description:Agonist activity at kappa opioid receptor in a [35S]GTPgammaS functional assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8.30nMAssay Description:Agonist activity at kappa opioid receptor in a [35S]GTPgammaS functional assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.40nMAssay Description:Agonist activity at kappa opioid receptor in a [35S]GTPgammaS functional assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30nMAssay Description:Agonist activity at kappa opioid receptor in a [35S]GTPgammaS functional assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.270nMAssay Description:Agonist activity at kappa opioid receptor in a [35S]GTPgammaS functional assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.490nMAssay Description:Agonist activity at kappa opioid receptor in a [35S]GTPgammaS functional assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.80nMAssay Description:Agonist activity at kappa opioid receptor in a [35S]GTPgammaS functional assayMore data for this Ligand-Target Pair
Affinity DataEC50: 24nMAssay Description:Agonist activity at kappa opioid receptor in a [35S]GTPgammaS functional assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0500nMAssay Description:Agonist activity at kappa opioid receptor in a [35S]GTPgammaS functional assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.420nMAssay Description:Agonist activity at kappa opioid receptor in a [35S]GTPgammaS functional assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.580nMAssay Description:Agonist activity at kappa opioid receptor in a [35S]GTPgammaS functional assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.520nMAssay Description:Agonist activity at kappa opioid receptor in a [35S]GTPgammaS functional assayMore data for this Ligand-Target Pair