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Found 24 Enz. Inhib. hit(s) with all data for entry = 50020319
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212403((1R,2R)-2-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,...)
Affinity DataEC50:  2.30nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212427(2-(3-(1-isopropyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  5nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212407((Z)-3-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  39.1nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212408(2-(3-(1,4,4,6-tetramethyl-2-oxo-1,2,3,4-tetrahydro...)
Affinity DataEC50:  144nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212409((1R,2R)-2-(3-(1-isopropyl-4,4,6-trimethyl-2-oxo-1,...)
Affinity DataEC50:  10nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212414(3-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetrah...)
Affinity DataEC50:  760nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212404(2-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetrah...)
Affinity DataEC50:  19.2nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212415(3-(3-(1-isopropyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  36.5nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212412(3-(3-(1-isopropyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  361nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212418(3-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetrah...)
Affinity DataEC50:  7.20nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212417(3-(4-(trifluoromethoxy)-3-(4,4,6-trimethyl-2-oxo-1...)
Affinity DataEC50:  1.40nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212274(5-((3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetra...)
Affinity DataEC50:  0.900nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212419(3-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetrah...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212411(3-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetrah...)
Affinity DataEC50:  37.7nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212277((E)-3-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  1.80nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212413((1S,2S)-2-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,...)
Affinity DataEC50:  361nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212423(3-(3-(1,4,4,6-tetramethyl-2-oxo-1,2,3,4-tetrahydro...)
Affinity DataEC50:  45.9nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212410(4-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetrah...)
Affinity DataEC50:  527nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212416((1S,2S)-2-(3-(1-isopropyl-4,4,6-trimethyl-2-oxo-1,...)
Affinity DataEC50:  198nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212406(3-(3-(1-isopropyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  3.40nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212422(2-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetrah...)
Affinity DataEC50:  116nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212426(3-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetrah...)
Affinity DataEC50:  27.9nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212425(2-(3-(1-isopropyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  208nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212405(3-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetrah...)
Affinity DataEC50:  70.2nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed