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Found 10 Enz. Inhib. hit(s) with all data for entry = 50046769
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50130404(CHEMBL3633687)
Affinity DataIC50:  8nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM5875(2-Anilino-5-aryloxazole 39 | N-[5-(Ethylsulfonyl)-...)
Affinity DataIC50:  22nMAssay Description:Inhibition of GST-tagged human recombinant VEGFR2 kinase expressed in Sf9 insect cells by radiometric protein kinase assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)
Affinity DataIC50:  39nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50130405(CHEMBL3633688)
Affinity DataIC50:  45nMAssay Description:Inhibition of His6-tagged KDR 789 to 1354 residues (unknown origin) using biotin-Ahx-AEEEYFFLA-amide substrate incubated for 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50130403(CHEMBL3633689)
Affinity DataIC50:  49nMAssay Description:Inhibition of GST-tagged human KDR expressed in Sf21 cells using 4:1 polyglutamic acid/tyrosine substrate incubated for 15 mins by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50130408(CHEMBL3633692)
Affinity DataIC50:  6.96E+3nMAssay Description:Inhibition of GST-tagged human recombinant VEGFR2 kinase expressed in Sf9 insect cells by radiometric protein kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50130410(CHEMBL3633690)
Affinity DataIC50:  4.01E+4nMAssay Description:Inhibition of GST-tagged human recombinant VEGFR2 kinase expressed in Sf9 insect cells by radiometric protein kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50130406(CHEMBL3633696)
Affinity DataIC50:  4.20E+4nMAssay Description:Inhibition of GST-tagged human recombinant VEGFR2 kinase expressed in Sf9 insect cells by radiometric protein kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50130407(CHEMBL3633695)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of GST-tagged human recombinant VEGFR2 kinase expressed in Sf9 insect cells by radiometric protein kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50130409(CHEMBL3633691)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of GST-tagged human recombinant VEGFR2 kinase expressed in Sf9 insect cells by radiometric protein kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed