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Found 24 Enz. Inhib. hit(s) with all data for entry = 50029139
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataIC50:  0.0800nMAssay Description:The compound was tested for its activity to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281730(4-Chloro-N-((S)-1-methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50:  0.390nMAssay Description:The compound was tested for its activity to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50006878((R)-1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  2nMpH: 6.5Assay Description:The compound was tested for its activity to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type B receptor in guinea pig brain at a pH of 6.5More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281732(4-Chloro-N-((R)-1-methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50:  2.90nMAssay Description:The compound was tested for its activity to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50061220(1-((S)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  3nMAssay Description:The compound was tested for its activity to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50060321(1H-Indole-2-carboxylic acid ((R)-1-methyl-2-oxo-5-...)
Affinity DataIC50:  8.30nMAssay Description:The compound was tested for its activity to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281729((4R,5S)-3-Oxo-4,5-diphenyl-pyrazolidine-1-carbothi...)
Affinity DataIC50:  17nMAssay Description:The compound was tested for its activity to inhibit the binding of [3H]-L-364,718 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50092155((4S,5R)-3-Oxo-4,5-diphenyl-pyrazolidine-1-carboxyl...)
Affinity DataIC50:  19nMpH: 7.4Assay Description:The compound was tested for its activity to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type B receptor in mouse brain at a pH of 6.5More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50092155((4S,5R)-3-Oxo-4,5-diphenyl-pyrazolidine-1-carboxyl...)
Affinity DataIC50:  31nMpH: 6.5Assay Description:The compound was tested for its activity to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type B receptor in mouse brain at a pH of 7.4More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281729((4R,5S)-3-Oxo-4,5-diphenyl-pyrazolidine-1-carbothi...)
Affinity DataIC50:  42nMAssay Description:The compound was tested for its activity to inhibit the binding of [3H]-L-364,718 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50061220(1-((S)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  150nMpH: 6.5Assay Description:The compound was tested for its activity to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type B receptor in guinea pig brain at a pH of 6.5More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataIC50:  270nMpH: 6.5Assay Description:The compound was tested for its activity to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type B receptor in guinea pig brain at a pH of 6.5More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50006878((R)-1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  280nMAssay Description:The compound was tested for its activity to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50092157((4R,5S)-3-Oxo-4,5-diphenyl-pyrazolidine-1-carboxyl...)
Affinity DataIC50:  370nMpH: 7.4Assay Description:The compound was tested for its activity to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type B receptor in mouse brain at a pH of 6.5More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50281731((4S,5R)-3-Oxo-4,5-diphenyl-pyrazolidine-1-carbothi...)
Affinity DataIC50:  550nMpH: 7.4Assay Description:The compound was tested for its activity to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type B receptor in mouse brain at a pH of 7.4More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281731((4S,5R)-3-Oxo-4,5-diphenyl-pyrazolidine-1-carbothi...)
Affinity DataIC50:  810nMAssay Description:The compound was tested for its activity to inhibit the binding of [3H]-L-364,718 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50281729((4R,5S)-3-Oxo-4,5-diphenyl-pyrazolidine-1-carbothi...)
Affinity DataIC50:  880nMpH: 7.4Assay Description:The compound was tested for its activity to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type B receptor in mouse brain at a pH of 7.4More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50281729((4R,5S)-3-Oxo-4,5-diphenyl-pyrazolidine-1-carbothi...)
Affinity DataIC50:  1.90E+3nMpH: 7.4Assay Description:The compound was tested for its activity to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type B receptor in mouse brain at a pH of 6.5More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281730(4-Chloro-N-((S)-1-methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50:  2.90E+3nMpH: 6.5Assay Description:The compound was tested for its activity to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type B receptor in guinea pig brain at a pH of 6.5More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50060321(1H-Indole-2-carboxylic acid ((R)-1-methyl-2-oxo-5-...)
Affinity DataIC50:  3.70E+3nMpH: 6.5Assay Description:The compound was tested for its activity to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type B receptor in guinea pig brain at a pH of 6.5More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50092157((4R,5S)-3-Oxo-4,5-diphenyl-pyrazolidine-1-carboxyl...)
Affinity DataIC50:  6.40E+3nMAssay Description:The compound was tested for its activity to inhibit the binding of [3H]-L-364,718 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281732(4-Chloro-N-((R)-1-methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50:  1.10E+4nMpH: 6.5Assay Description:The compound was tested for its activity to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type B receptor in guinea pig brain at a pH of 6.5More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50092155((4S,5R)-3-Oxo-4,5-diphenyl-pyrazolidine-1-carboxyl...)
Affinity DataIC50:  1.16E+4nMAssay Description:The compound was tested for its activity to inhibit the binding of [3H]-L-364,718 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50092155((4S,5R)-3-Oxo-4,5-diphenyl-pyrazolidine-1-carboxyl...)
Affinity DataIC50:  2.05E+4nMAssay Description:The compound was tested for its activity to inhibit the binding of [3H]-L-364,718 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article