Compile Data Set for Download or QSAR
maximum 50k data
Found 33 Enz. Inhib. hit(s) with all data for entry = 50031320
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311121(CHEMBL1079108 | N-(4-(2-amino-2-methylpropyl)pheny...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311117(CHEMBL1078900 | N-(4-(2-amino-2-methylpropyl)pheny...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311092((S)-4-(3-hexylureido)-N-(4-(2-(2-hydroxy-3-(4-hydr...)
Affinity DataIC50:  13nMAssay Description:Displacement of [35S]MK0677 from human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311116(CHEMBL1078899 | N-(4-(2-amino-2-methylpropyl)pheny...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311119(CHEMBL1079091 | N-(4-(2-amino-2-methylpropyl)pheny...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311120(CHEMBL1079107 | N-(4-(2-amino-2-methylpropyl)pheny...)
Affinity DataIC50:  21nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311118(CHEMBL1078982 | N-(4-(2-amino-2-methylpropyl)pheny...)
Affinity DataIC50:  28nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311096(CHEMBL1079046 | N-(4-(2-(ethylamino)-2-methylpropy...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311092((S)-4-(3-hexylureido)-N-(4-(2-(2-hydroxy-3-(4-hydr...)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at human GHS-R1a expressed in HEK293 cells assessed as inhibition of ghrelin-stimulated intracellular calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311095(CHEMBL1079045 | N-(4-(2-amino-2-methylpropyl)pheny...)
Affinity DataIC50:  46nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311114(CHEMBL1078700 | N-(4-(2-amino-2-methylpropyl)pheny...)
Affinity DataIC50:  69nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311115(CHEMBL1078960 | N-(4-(2-amino-2-methylpropyl)pheny...)
Affinity DataIC50:  77nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311109(CHEMBL1078497 | N-(4-(2-amino-2-methylpropyl)pheny...)
Affinity DataIC50:  97nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311098(CHEMBL1079872 | N-(4-(3-aminopropyl)phenyl)-4-(3-h...)
Affinity DataIC50:  108nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311111(CHEMBL1078608 | N-(4-(2-amino-2-methylpropyl)pheny...)
Affinity DataIC50:  128nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311112(CHEMBL1078677 | N-(4-(2-amino-2-methylpropyl)pheny...)
Affinity DataIC50:  138nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311113(CHEMBL1078699 | N-(4-(2-amino-2-methylpropyl)pheny...)
Affinity DataIC50:  161nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311108(CHEMBL1078403 | N-(4-(2-amino-2-methylpropyl)pheny...)
Affinity DataIC50:  241nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311110(CHEMBL1078498 | N-(4-(2-amino-2-methylpropyl)pheny...)
Affinity DataIC50:  263nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311094(CHEMBL1077839 | N-(4-(2-aminoethyl)phenyl)-4-(3-he...)
Affinity DataIC50:  272nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311099(CHEMBL1079873 | N-(4-(3-amino-3-methylbutyl)phenyl...)
Affinity DataIC50:  310nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311102(CHEMBL1079302 | N-(3-(3-aminopropyl)phenyl)-4-(3-h...)
Affinity DataIC50:  429nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311100(CHEMBL1082044 | N-(4-(3-amino-2,2-dimethylpropyl)p...)
Affinity DataIC50:  444nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311107(CHEMBL1078402 | N-(4-(2-amino-2-methylpropyl)pheny...)
Affinity DataIC50:  474nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311101(CHEMBL1079340 | N-(3-(2-aminoethyl)phenyl)-4-(3-he...)
Affinity DataIC50:  625nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311103(4-(3-hexylureido)-N-(4-(2-methyl-2-(2,2,2-trifluor...)
Affinity DataIC50:  682nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311106(CHEMBL1078115 | N-(4-(2-amino-2-methylpropyl)pheny...)
Affinity DataIC50:  846nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311105(CHEMBL1078114 | N-(4-(2-amino-2-methylpropyl)pheny...)
Affinity DataIC50:  1.65E+3nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311097(CHEMBL1078533 | N-(4-(aminomethyl)phenyl)-4-(3-hex...)
Affinity DataIC50:  1.72E+3nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311093(4-(3-hexylureido)-N-phenylbenzenesulfonamide | CHE...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311095(CHEMBL1079045 | N-(4-(2-amino-2-methylpropyl)pheny...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of human adrenergic beta3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311104(CHEMBL1079323 | N-(4-(2-amino-2-methylpropyl)pheny...)
Affinity DataIC50:  5.62E+3nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311095(CHEMBL1079045 | N-(4-(2-amino-2-methylpropyl)pheny...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human adrenergic beta3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed