Compile Data Set for Download or QSAR
maximum 50k data
Found 23 Enz. Inhib. hit(s) with all data for entry = 50048373
LigandPNGBDBM50213779(CHEMBL313598)
Affinity DataIC50:  0.0200nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213592(CHEMBL315236)
Affinity DataIC50:  0.0400nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213695(CHEMBL89032)
Affinity DataIC50:  0.0400nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213685(CHEMBL431853)
Affinity DataIC50:  0.0600nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213687(CHEMBL87244)
Affinity DataIC50:  0.0700nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213697(CHEMBL84908)
Affinity DataIC50:  0.0700nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213687(CHEMBL87244)
Affinity DataIC50:  0.0700nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213593(CHEMBL91046)
Affinity DataIC50:  0.0800nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213688(CHEMBL86538)
Affinity DataIC50:  0.0800nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213782(CHEMBL264304)
Affinity DataIC50:  0.0800nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213680(CHEMBL87091)
Affinity DataIC50:  0.0900nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213681(CHEMBL433010)
Affinity DataIC50:  0.0900nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213591(CHEMBL84795)
Affinity DataIC50:  0.100nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213783(CHEMBL328985)
Affinity DataIC50:  0.100nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213679(5-Beta-Ketosulfoxide Imidazolyl Biphenyl Sulfonylu...)
Affinity DataIC50:  0.200nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213781(CHEMBL327927)
Affinity DataIC50:  0.200nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213594(CHEMBL85075)
Affinity DataIC50:  0.300nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213682(CHEMBL91047)
Affinity DataIC50:  0.300nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213778(CHEMBL312990)
Affinity DataIC50:  0.300nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213780(CHEMBL316402)
Affinity DataIC50:  0.350nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50031530(2-Butyl-4-(methylthio)-1-[[2'-[[[(propylamino)carb...)
Affinity DataIC50:  0.5nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213684(CHEMBL89772)
Affinity DataIC50:  1.80nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50285756(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  3.80nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails