Compile Data Set for Download or QSAR
maximum 50k data
Found 48 Enz. Inhib. hit(s) with all data for entry = 50031983
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM13065(5-(4-chlorophenyl)-1-(4-methoxyphenyl)-3-(trifluor...)
Affinity DataIC50:  10nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50029593(CHEMBL7162 | N-(2-(cyclohexyloxy)-4-nitrophenyl)me...)
Affinity DataIC50:  150nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322764(CHEMBL1171447 | clematernoside K)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322755(3-O-alpha-L-rhamnopyranosyl-(1-6)-[beta-D-glucopyr...)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322755(3-O-alpha-L-rhamnopyranosyl-(1-6)-[beta-D-glucopyr...)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322754(3-O-beta-Dglucopyranosyl-(1-2)-alpha-L-rhamnopyran...)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322764(CHEMBL1171447 | clematernoside K)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322758(3-O-[(6-O-isoferuloyl)-beta-D-glucopyranosyl]-(1-4...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322759(3-O-beta-D-glucopyranosyl-(1-3)-[(2-O-isoferuloyl)...)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322761(CHEMBL1171258 | clematernoside C)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322760(CHEMBL1171257 | clematernoside B)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322758(3-O-[(6-O-isoferuloyl)-beta-D-glucopyranosyl]-(1-4...)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322756(3-O-[(3-O-isoferuloyl)-beta-D-glucopyranosyl]-(1-4...)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322754(3-O-beta-Dglucopyranosyl-(1-2)-alpha-L-rhamnopyran...)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322757(3-O-[(6-O-isoferuloyl)-beta-D-glucopyranosyl]-(1-4...)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322760(CHEMBL1171257 | clematernoside B)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322763(CHEMBL1171446 | clematernoside E)
Affinity DataIC50:  8.30E+3nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322763(CHEMBL1171446 | clematernoside E)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322762(CHEMBL1171445 | clematernoside D)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322756(3-O-[(3-O-isoferuloyl)-beta-D-glucopyranosyl]-(1-4...)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322761(CHEMBL1171258 | clematernoside C)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322757(3-O-[(6-O-isoferuloyl)-beta-D-glucopyranosyl]-(1-4...)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322759(3-O-beta-D-glucopyranosyl-(1-3)-[(2-O-isoferuloyl)...)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322762(CHEMBL1171445 | clematernoside D)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322745(CHEMBL1171452 | clematichinenoside C)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322746(CHEMBL1171453 | clematichinenoside B)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322747(CHEMBL1171451 | huzhangoside D)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322748(CHEMBL1171450 | huzhangoside B)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322749(CHEMBL1171449 | kizuta saponin K12)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50259663(3beta-O-[alpha-L-rhamnopyranosyl-(1->2)alpha-L-ara...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322750(3beta-[(alpha-L-arabinopyranosyl)oxy]-23-hydroxyol...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322751(CHEMBL1171250 | ciwujianoside C3)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322752(3beta,23-dihydroxyolean-12-en-28-oic acid O-alpha-...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322753(CHEMBL1171448 | cirensenoside O)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322748(CHEMBL1171450 | huzhangoside B)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322753(CHEMBL1171448 | cirensenoside O)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322746(CHEMBL1171453 | clematichinenoside B)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322744(CHEMBL1171454 | clematomandshurica saponin C)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322750(3beta-[(alpha-L-arabinopyranosyl)oxy]-23-hydroxyol...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322749(CHEMBL1171449 | kizuta saponin K12)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322744(CHEMBL1171454 | clematomandshurica saponin C)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322752(3beta,23-dihydroxyolean-12-en-28-oic acid O-alpha-...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322765(3-O-beta-D-glucopyranosyl-(1-4)-beta-D-glucopyrano...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50259663(3beta-O-[alpha-L-rhamnopyranosyl-(1->2)alpha-L-ara...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322751(CHEMBL1171250 | ciwujianoside C3)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322747(CHEMBL1171451 | huzhangoside D)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322765(3-O-beta-D-glucopyranosyl-(1-4)-beta-D-glucopyrano...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX2 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50322745(CHEMBL1171452 | clematichinenoside C)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of COX1 by microplate readerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed