Affinity DataIC50: 0.0230nMAssay Description:Antagonist activity at alpha2bbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:Antagonist activity at alphavbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Antagonist activity at alphavbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Antagonist activity at alpha2bbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.190nMAssay Description:Antagonist activity at alphavbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.210nMAssay Description:Antagonist activity at alpha2bbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.230nMAssay Description:Antagonist activity at alphavbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.25nMAssay Description:Antagonist activity at alphavbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at alphavbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.360nMAssay Description:Antagonist activity at alphavbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at alpha2bbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.440nMAssay Description:Antagonist activity at alphavbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.440nMAssay Description:Antagonist activity at alpha2bbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.480nMAssay Description:Antagonist activity at alphavbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.560nMAssay Description:Antagonist activity at alpha2bbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.770nMAssay Description:Antagonist activity at alphavbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.780nMAssay Description:Antagonist activity at alpha2bbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.940nMAssay Description:Antagonist activity at alpha2bbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.980nMAssay Description:Antagonist activity at alpha2bbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at alpha2bbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at alphavbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Antagonist activity at alpha2bbeta3 integrin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Antagonist activity at alphavbeta3 integrin receptor human VSMC assessed as inhibition of vitronectin-induced cell adhesionMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Antagonist activity at alphavbeta3 integrin receptor human VSMC assessed as inhibition of vitronectin-induced cell adhesionMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Antagonist activity at alphavbeta3 integrin receptor human VSMC assessed as inhibition of vitronectin-induced cell adhesionMore data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Antagonist activity at alphavbeta3 integrin receptor human VSMC assessed as inhibition of vitronectin-induced cell adhesionMore data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:Antagonist activity at alphavbeta3 integrin receptor human VSMC assessed as inhibition of vitronectin-induced cell adhesionMore data for this Ligand-Target Pair
Affinity DataIC50: 72nMAssay Description:Antagonist activity at alphavbeta3 integrin receptor human VSMC assessed as inhibition of vitronectin-induced cell adhesionMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Antagonist activity at alphavbeta3 integrin receptor human VSMC assessed as inhibition of vitronectin-induced cell adhesionMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Antagonist activity at alphavbeta3 integrin receptor human VSMC assessed as inhibition of vitronectin-induced cell adhesionMore data for this Ligand-Target Pair
Affinity DataIC50: 390nMAssay Description:Antagonist activity at alphavbeta3 integrin receptor human VSMC assessed as inhibition of vitronectin-induced cell adhesionMore data for this Ligand-Target Pair
Affinity DataIC50: 530nMAssay Description:Antagonist activity at alphavbeta3 integrin receptor human VSMC assessed as inhibition of vitronectin-induced cell adhesionMore data for this Ligand-Target Pair
Affinity DataIC50: 660nMAssay Description:Antagonist activity at alphavbeta3 integrin receptor human VSMC assessed as inhibition of vitronectin-induced cell adhesionMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at AhR in human MCF-7 cells assessed as increase of CYP1A1-dependent 7-ethoxyresorufin O-deethylase activityMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at AhR in human MCF-7 cells assessed as increase of CYP1A1-dependent 7-ethoxyresorufin O-deethylase activityMore data for this Ligand-Target Pair
Affinity DataEC50: 330nMAssay Description:Agonist activity at AhR in human MCF-7 cells assessed as increase of CYP1A1-dependent 7-ethoxyresorufin O-deethylase activityMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonist activity at AhR in human MCF-7 cells assessed as increase of CYP1A1-dependent 7-ethoxyresorufin O-deethylase activityMore data for this Ligand-Target Pair
Affinity DataEC50: 270nMAssay Description:Agonist activity at AhR in human MCF-7 cells assessed as increase of CYP1A1-dependent 7-ethoxyresorufin O-deethylase activityMore data for this Ligand-Target Pair
Affinity DataEC50: 450nMAssay Description:Agonist activity at AhR in human MCF-7 cells assessed as increase of CYP1A1-dependent 7-ethoxyresorufin O-deethylase activityMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataEC50: 170nMAssay Description:Partial agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Partial agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataEC50: 53nMAssay Description:Partial agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataEC50: 29nMAssay Description:Partial agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataEC50: 1.60nMAssay Description:Partial agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataEC50: 5.70nMAssay Description:Partial agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataEC50: 220nMAssay Description:Partial agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataEC50: 76nMAssay Description:Partial agonist activity at PPARdeltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The University Of Tokyo
Curated by ChEMBL
The University Of Tokyo
Curated by ChEMBL
Affinity DataEC50: 790nMAssay Description:Agonist activity at PPARalphaMore data for this Ligand-Target Pair